SCHEMBL28360752

SCHEMBL28360752

COc1ccccc1C=CC(=O)C=Cc1ccc(-c2cc(=O)oc3ccccc23)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 3/20 0.53
TFEB P19484 1/20 0.53
LY96 Q9Y6Y9 3/20 0.51
KDM4E B2RXH2 4/20 0.48
NPC1 O15118 2/20 0.48
MAPT P10636 2/20 0.48
RAB9A P51151 2/20 0.48
MAPK1 P28482 1/20 0.48
ATM Q13315 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
TUBB4A P04350 3/20 0.46
TUBB P07437 3/20 0.46
TUBA3C P0DPH7 3/20 0.46
TUBA1B P68363 3/20 0.46
TUBA4A P68366 3/20 0.46
TUBB4B P68371 3/20 0.46
TUBB3 Q13509 3/20 0.46
TUBB2A Q13885 3/20 0.46
TUBB8 Q3ZCM7 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28357068 0.90 ALDH1A1 (0.55) KDM4ENPC1MAPTRAB9AMAPK1
SCHEMBL28356950 0.89 TUBB4A (0.54) NFE2L2KDM4EMAPTRAB9AMAPK1
SCHEMBL28356915 0.87 NFE2L2 (0.58) NFE2L2TFEBLY96KDM4ENPC1
SCHEMBL28360755 0.85 CA9 (0.49) KDM4ENPC1MAPTRAB9ANPSR1
SCHEMBL28360775 0.84 HSD11B1 (0.50) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL28360863 0.82 F3 (0.50) KDM4ENPC1MAPTRAB9AMAPK1
SCHEMBL28356945 0.82 CA9 (0.53) NPC1MAPTRAB9ALMNAHPGD
SCHEMBL28357183 0.79 HSD11B1 (0.47) KDM4ETUBB4ATUBBTUBA3CTUBA1B
SCHEMBL28756580 0.78 F3 (0.56) KDM4ENPC1MAPTRAB9ANOD2
SCHEMBL28356957 0.78 ALDH1A1 (0.46) KDM4ENPC1MAPTRAB9ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106928176-B Coumarin-containing 1, 4-pentadiene-3-ketone derivative and preparation method and application thereof 贵州大学 2020-02-18 CN disclosed