SCHEMBL2837167

SCHEMBL2837167

NNC(=O)c1csc(Br)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.53
LMNA P02545 3/20 0.53
OGG1 O15527 1/20 0.48
KDM4E B2RXH2 6/20 0.46
MAPT P10636 4/20 0.44
L3MBTL1 Q9Y468 3/20 0.44
GAA P10253 3/20 0.44
BLM P54132 2/20 0.44
TDP1 Q9NUW8 2/20 0.44
HTT P42858 2/20 0.44
NSD2 O96028 1/20 0.44
ALPL P05186 1/20 0.44
POLB P06746 1/20 0.44
ALPI P09923 1/20 0.44
ALPG P10696 1/20 0.44
APEX1 P27695 1/20 0.44
RECQL P46063 1/20 0.44
CASP6 P55212 1/20 0.44
MPO P05164 2/20 0.41
CYP3A4 P08684 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1750114 0.80 HDAC8 (0.45) ALDH1A1LMNAMAPTL3MBTL1TDP1
SCHEMBL8631005 0.79 ALDH1A1 (0.37) ALDH1A1LMNAMAPTL3MBTL1TDP1
SCHEMBL7217724 0.79 L3MBTL1 (0.48) ALDH1A1LMNAMAPTL3MBTL1GAA
SCHEMBL25233005 0.78 HPGD (0.46) ALDH1A1KDM4EMAPTL3MBTL1GAA
SCHEMBL1674356 0.77
SCHEMBL26469193 0.77 GAA (0.56) ALDH1A1LMNAKDM4EMAPTL3MBTL1
SCHEMBL27682287 0.76 CES2 (0.39) ALDH1A1LMNATDP1RAB9ANPC1
SCHEMBL29450062 0.76 DAO (0.59) ALDH1A1LMNAOGG1KDM4EMAPT
SCHEMBL655351 0.76 DAO (0.59) ALDH1A1LMNAMAPTL3MBTL1TDP1
SCHEMBL20521778 0.74 SMYD3 (0.46) ALDH1A1MAPTL3MBTL1HTTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010065383-A1 CALCILYTIC COMPOUNDS GLAXOSMITHKLINE LLC (US) 2010-06-10 WO disclosed
WO-2010039913-A1 CALCILYTIC COMPOUNDS GLAXOSMITHKLINE LLC (US) 2010-04-08 WO disclosed