SCHEMBL8631005

SCHEMBL8631005

NP(N)(=O)NC(=O)c1csc(Br)c1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
RAB9A P51151 3/20 0.36
NPC1 O15118 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.31
MAPT P10636 1/20 0.31
MAPK1 P28482 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
HSD17B10 Q99714 1/20 0.31
CES2 O00748 1/20 0.31
CES1 P23141 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2837167 0.79 ALDH1A1 (0.53) ALDH1A1LMNARAB9ANPC1TDP1
SCHEMBL8631119 0.79 DAO (0.53) ALDH1A1LMNARAB9ANPC1TDP1
SCHEMBL8705579 0.79 DAO (0.53) ALDH1A1LMNARAB9ANPC1TDP1
SCHEMBL1750114 0.76 HDAC8 (0.45) ALDH1A1LMNARAB9ANPC1TDP1
SCHEMBL8628173 0.75 RAB9A (0.36) ALDH1A1LMNARAB9ANPC1TDP1
SCHEMBL10935869 0.74 KDM4E (0.38) ALDH1A1LMNATDP1MAPTL3MBTL1
SCHEMBL8630112 0.73 GAA (0.51) ALDH1A1RAB9ANPC1TDP1SMN1; SMN2
SCHEMBL8630018 0.73 ALDH1A1 (0.65) ALDH1A1LMNARAB9ANPC1TDP1
SCHEMBL1674356 0.72
SCHEMBL7217724 0.71 L3MBTL1 (0.48) ALDH1A1LMNARAB9ANPC1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5840917-A ADMINISTERING TO MAMMAL TO ERADICATE HELICOBACTER PYLORI TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-11-24 US disclosed
WO-1998042347-A1 PHARMACEUTICAL COMPOSITION CONTAINING A PHOSPHORYLAMIDE AND AN AYNTIBIOTIC TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-10-01 WO disclosed
EP-0852498-A1 PHOSPHORYLAMIDES, THEIR PREPARATION AND USE Takeda Chemical Industries, Ltd. (JP) 1998-07-15 EP disclosed
WO-1997011705-A1 PHOSPHORYLAMIDES, THEIR PREPARATION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-04-03 WO disclosed