SCHEMBL28378012

SCHEMBL28378012

O=C(N[C@@H]1CCCC[C@H]1c1cc(NC(=O)C(F)(F)F)n[nH]1)OCc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 1/20 0.46
CDK2 P24941 4/20 0.43
CCNA2 P20248 2/20 0.43
CCNA1 P78396 2/20 0.43
EPHX1 P07099 1/20 0.42
CASP3 P42574 3/20 0.41
TACR1 P25103 2/20 0.41
ALDH1A1 P00352 2/20 0.41
CTSL P07711 1/20 0.40
CTSB P07858 1/20 0.40
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
CCNE1 P24864 1/20 0.39
CDK9 P50750 1/20 0.39
CDK5 Q00535 1/20 0.39
CDK5R1 Q15078 1/20 0.39
CPB1 P15086 1/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22204486 0.83 CDK2 (0.40) CDK2CCNA2CCNA1CCNE1CDK9
SCHEMBL22204485 0.83 CDK2 (0.40) CDK2CCNA2CCNA1CCNE1CDK9
SCHEMBL28383571 0.82 CPB1 (0.46) EPHX1CASP3TACR1ALDH1A1CTSL
SCHEMBL29444919 0.81 HDAC4 (0.39) CDK2CCNA2CCNA1CCNE1CDK9
SCHEMBL29444920 0.81 HDAC4 (0.39) CDK2CCNA2CCNA1CCNE1CDK9
SCHEMBL28381708 0.76 FGFR4 (0.44) USP30EPHX1CASP3ALDH1A1CTSL
SCHEMBL28378015 0.73 ENPP2 (0.46) USP30CDK2CCNA2CCNA1EPHX1
SCHEMBL6612597 0.73 EPHX1 (0.63) EPHX1CASP3ALDH1A1CTSLCTSB
SCHEMBL22204505 0.72 CCNA2 (0.41) CDK2CCNA2CCNA1
Trifluoroacetic Acid SCHEMBL5029718 0.71 ALDH1A1 (0.52) EPHX1CASP3TACR1ALDH1A1CTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110997637-B Aromatic derivative, preparation method and application thereof in medicine 保仕健生物科技(上海)有限公司 2022-09-27 CN disclosed
CN-110997637-A Aromatic derivative, preparation method and application thereof in medicine 博奥阿迪斯生物科技公司 2020-04-10 CN disclosed