SCHEMBL28387604

SCHEMBL28387604

CC(C)(C)OC(=O)NNC(=O)c1ccnc(N)n1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.40
MEN1 O00255 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40
NUDT1 P36639 4/20 0.39
ATR Q13535 1/20 0.38
GSK3A P49840 1/20 0.38
GSK3B P49841 1/20 0.38
ROCK1 Q13464 1/20 0.36
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36
APLNR P35414 1/20 0.35
IRAK4 Q9NWZ3 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.34
MAPKAPK2 P49137 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1029794 0.79 NUDT1 (0.42) GAANUDT1ATRROCK1KDM4E
SCHEMBL18038254 0.74 DYRK1A (0.44) GSK3BLMNAIRAK4ALDH1A1
SCHEMBL16572967 0.74 PTPN11 (0.45) NUDT1GSK3AGSK3BROCK1KDM4E
SCHEMBL107631 0.73 GRM4 (0.45) GAAMEN1NPC1RAB9AKMT2A
SCHEMBL106399 0.72 GAA (0.40) GAAMEN1NPC1RAB9AKMT2A
SCHEMBL8281629 0.72 TRPA1 (0.46) GAAMEN1NPC1RAB9AKMT2A
SCHEMBL106420 0.72 APLNR (0.50) GAAMEN1NPC1RAB9AKMT2A
SCHEMBL1789196 0.71 ROCK1 (0.55) GAANPC1RAB9AROCK1KDM4E
SCHEMBL12579446 0.70 TRPA1 (0.44) GAAMEN1NPC1RAB9AKMT2A
SCHEMBL3336071 0.70 HRH4 (0.60) NUDT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115504986-B Apoptosis signal regulating kinase inhibitor and preparation method and application thereof 江苏豪森药业集团有限公司 2024-05-14 CN disclosed
CN-115504986-A Apoptosis signal regulating kinase inhibitor and preparation method and application thereof 江苏豪森药业集团有限公司 2022-12-23 CN disclosed
CN-111094250-B Apoptosis signal regulating kinase inhibitor and preparation method and application thereof 江苏豪森药业集团有限公司 2022-11-04 CN disclosed
CN-111094250-A Apoptosis signal regulating kinase inhibitor and preparation method and application thereof 江苏豪森药业集团有限公司 2020-05-01 CN disclosed