SCHEMBL2839722

SCHEMBL2839722

Cc1nc(-c2ncccc2OCc2ccccc2)n(CCc2ccccc2)c(=O)c1Br

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 5/20 0.46
ALDH1A1 P00352 4/20 0.46
CYP1A2 P05177 4/20 0.46
CYP2C9 P11712 3/20 0.46
CYP2C19 P33261 3/20 0.46
CYP3A4 P08684 3/20 0.46
LMNA P02545 2/20 0.46
HIF1A Q16665 1/20 0.46
CASR P41180 6/20 0.45
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
MAPK14 Q16539 5/20 0.40
USP2 O75604 2/20 0.40
CYP2D6 P10635 1/20 0.39
LTA4H P09960 1/20 0.39
GFER P55789 1/20 0.39
NR1I2 O75469 1/20 0.39
GRM5 P41594 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4145053 0.87 CASR (0.57) TSHRALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL2840670 0.85 HTR2C (0.40) MAPK14LTA4HGRM5
SCHEMBL2839694 0.84 CYP1A2 (0.43) TSHRALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL2837296 0.83 CASR (0.49) TSHRALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL2838847 0.83 CASR (0.55) TSHRALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL4138596 0.82 CASR (0.51) TSHRALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL2838115 0.81 CASR (0.55) TSHRALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL2835830 0.78 CASR (0.66) TSHRALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL13851597 0.77 CASR (0.58) TSHRALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL4138763 0.77 CASR (0.63) TSHRALDH1A1LMNACASRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010039913-A1 CALCILYTIC COMPOUNDS GLAXOSMITHKLINE LLC (US) 2010-04-08 WO disclosed