SCHEMBL28398159

SCHEMBL28398159

Cc1cn(CC2CCN(C(=O)OC(C)(C)C)CC2)c(=O)nc1N

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 2/20 0.50
KDM4E B2RXH2 2/20 0.43
PKM P14618 1/20 0.43
CTSD P07339 1/20 0.42
CTSE P14091 1/20 0.42
TGFBR1 P36897 1/20 0.42
FAAH O00519 1/20 0.42
TP53 P04637 1/20 0.41
GPR119 Q8TDV5 7/20 0.41
FPR2 P25090 1/20 0.41
MAPT P10636 1/20 0.41
THRB P10828 1/20 0.41
PIK3CA P42336 1/20 0.41
PRKDC P78527 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28398168 0.88 BACE1 (0.49) BACE1KDM4EPKMCTSDCTSE
SCHEMBL28402009 0.81 BACE1 (0.51) BACE1KDM4EPKMCTSDCTSE
SCHEMBL17406871 0.79 BACE1 (0.42) BACE1KDM4EPKMTGFBR1FAAH
SCHEMBL15645613 0.76 BACE1 (0.48) BACE1KDM4EPKMTGFBR1FAAH
SCHEMBL17406877 0.75 TGFBR1 (0.44) KDM4EPKMTGFBR1FAAHGPR119
SCHEMBL948973 0.74 GPR119 (0.50) BACE1KDM4EPKMFAAHGPR119
SCHEMBL22650836 0.74 BACE1 (0.48) BACE1KDM4EPKMGPR119FPR2
SCHEMBL28401089 0.74 PI4KA (0.51) BACE1TGFBR1GPR119
SCHEMBL17394767 0.74 TGFBR1 (0.43) KDM4EPKMTGFBR1FAAHGPR119
SCHEMBL4771557 0.73 BACE1 (0.51) BACE1KDM4EPKMFAAHGPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106883217-B Nucleoside base hydroxamic acid derivative compound and preparation method and application thereof 清华大学深圳研究生院 2020-05-22 CN disclosed