SCHEMBL28401656

SCHEMBL28401656

Cn1ccnc1-c1cc2ccccc2[nH]1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.51
HSD17B10 Q99714 2/20 0.51
CASP1 P29466 1/20 0.51
CASP7 P55210 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
AURKA O14965 1/20 0.48
AURKB Q96GD4 1/20 0.48
GSK3B P49841 1/20 0.47
RAB9A P51151 4/20 0.46
NPC1 O15118 3/20 0.46
ITK Q08881 4/20 0.46
ESR1 P03372 2/20 0.46
CYP19A1 P11511 1/20 0.45
PARP1 P09874 1/20 0.45
MAPT P10636 4/20 0.43
MEN1 O00255 3/20 0.43
ALDH1A1 P00352 3/20 0.43
HPGD P15428 3/20 0.43
KMT2A Q03164 3/20 0.43
USP2 O75604 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6406795 0.79 GSK3B (0.44) KDM4EHSD17B10AURKAAURKBGSK3B
SCHEMBL28405187 0.79 PARP1 (0.52) KDM4EHSD17B10AURKAAURKBGSK3B
SCHEMBL17680533 0.78 AURKA (0.48) KDM4EHSD17B10AURKAAURKBGSK3B
SCHEMBL693581 0.76 GSK3B (0.59) KDM4EHSD17B10AURKAAURKBGSK3B
SCHEMBL17680257 0.73 COMT (0.49) KDM4EHSD17B10AURKAAURKBGSK3B
SCHEMBL14077039 0.73 PARP1 (0.49) KDM4EHSD17B10AURKAAURKBGSK3B
SCHEMBL30693865 0.73 KDM4E (0.68) KDM4EHSD17B10CASP1CASP7L3MBTL1
SCHEMBL374022 0.71 RAB9A (0.74) KDM4EHSD17B10AURKAAURKBGSK3B
SCHEMBL29631691 0.71 RAB9A (0.74) KDM4EHSD17B10AURKAAURKBGSK3B
SCHEMBL21318393 0.71 PDGFRB (0.52) KDM4EHSD17B10L3MBTL1AURKAAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111225915-B Imidazopyridine compounds as PAD inhibitors 朱比兰特埃皮帕德有限公司 2023-03-07 CN disclosed
CN-111225915-A Imidazopyridine compounds as PAD inhibitors 朱比兰特埃皮帕德有限公司 2020-06-02 CN disclosed