SCHEMBL28406243

SCHEMBL28406243

COc1cccc(-c2cn(S(=O)(=O)c3ccc(C)cc3)nn2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.47
NFE2L2 Q16236 1/20 0.47
POLB P06746 1/20 0.47
STIM1 Q13586 1/20 0.45
ORAI1 Q96D31 1/20 0.45
MAPT P10636 5/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA5A P35218 1/20 0.44
CA5B Q9Y2D0 1/20 0.44
TP53 P04637 3/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
HSD17B10 Q99714 2/20 0.44
ALDH1A1 P00352 2/20 0.44
KDM4E B2RXH2 1/20 0.44
NPC1 O15118 1/20 0.44
HPGD P15428 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26252983 0.86 CA2 (0.57) KEAP1NFE2L2MAPTCA1CA2
SCHEMBL30938679 0.86 CA2 (0.57) KEAP1NFE2L2MAPTCA1CA2
SCHEMBL28396678 0.85 KMT2A (0.55) MAPTCA1CA2CA5ACA5B
SCHEMBL28401134 0.83 CA1 (0.46) MAPTCYP3A4CYP2C9CYP2C19CA1
SCHEMBL28888736 0.83 GRM5 (0.46) KEAP1NFE2L2POLBMAPTCYP3A4
SCHEMBL30938684 0.83 CA1 (0.46) MAPTCYP3A4CYP2C9CYP2C19CA1
SCHEMBL28400475 0.83 MAPT (0.46) KEAP1NFE2L2MAPTCYP3A4CYP2C9
SCHEMBL29710495 0.82 STIM1 (0.50) KEAP1NFE2L2STIM1ORAI1MAPT
SCHEMBL28562832 0.82 STIM1 (0.50) KEAP1NFE2L2STIM1ORAI1MAPT
SCHEMBL22558313 0.82 MAPT (0.56) MAPTCA1CA2CA5ACA5B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111170955-B Green preparation method of 2H-1,2,3-triazole compound 河南师范大学 2023-04-07 CN disclosed
CN-111170955-A Green preparation method of 2H-1,2, 3-triazole compound 河南师范大学 2020-05-19 CN disclosed