SCHEMBL28409481

SCHEMBL28409481

COc1ccc(-c2cc3ccc(Cl)cc3o2)cc1OC

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 2/20 0.54
ABCB1 P08183 4/20 0.52
ABCG2 Q9UNQ0 3/20 0.52
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
TP53 P04637 1/20 0.52
MDM2 Q00987 1/20 0.52
CALCRL Q16602 1/20 0.51
CA1 P00915 2/20 0.50
CA2 P00918 2/20 0.50
MAPK1 P28482 2/20 0.50
HSD17B10 Q99714 2/20 0.50
MAPT P10636 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
CSNK2A2 P19784 1/20 0.50
CSNK2B P67870 1/20 0.50
CSNK2A1 P68400 1/20 0.50
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 1/20 0.50
GLA P06280 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16011311 0.85 ABCB1 (0.66) PDE4AABCB1ABCG2MEN1KMT2A
SCHEMBL20147031 0.82 CALCRL (0.74) PDE4AABCB1ABCG2MEN1KMT2A
SCHEMBL28409862 0.82 PDE4A (0.54) PDE4AABCB1ABCG2MEN1KMT2A
SCHEMBL11733704 0.82 KCNA5 (0.62) ABCG2MEN1KMT2ATP53CA1
SCHEMBL11672469 0.80 ABCB1 (0.65) PDE4AABCB1ABCG2MEN1KMT2A
SCHEMBL21860285 0.78 ALOX5 (0.52) PDE4AABCB1ABCG2MEN1KMT2A
SCHEMBL27908290 0.78 CSNK2A2 (0.80) ABCB1ABCG2MEN1KMT2ATP53
SCHEMBL28407601 0.75 PDE4A (0.53) PDE4AABCB1ABCG2MEN1KMT2A
SCHEMBL25824711 0.75 CYP2A6 (0.52) CA1CA2SMN1; SMN2CYP1B1CYP1A1
SCHEMBL19887207 0.74 GABRP (0.58) CYP1B1CYP1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107325067-B Mulberry octyl element M derivative of phosphodiesterase 4 inhibitor and application thereof 广州中医药大学 2020-05-12 CN claimed
CN-107325067-B Mulberry octyl element M derivative of phosphodiesterase 4 inhibitor and application thereof 广州中医药大学 2020-05-12 CN disclosed