SCHEMBL28413243

SCHEMBL28413243

O=C1CCC(c2ccccc2)N1O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.49
CHRM2 P08172 1/20 0.47
CHRM4 P08173 1/20 0.47
CHRM5 P08912 1/20 0.47
CHRM1 P11229 1/20 0.47
CHRM3 P20309 1/20 0.47
SRD5A1 P18405 1/20 0.46
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
KDM4E B2RXH2 2/20 0.41
CYP3A4 P08684 1/20 0.41
THRB P10828 1/20 0.41
TSHR P16473 1/20 0.41
THPO P40225 1/20 0.41
MAPK1 P28482 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
HTT P42858 1/20 0.41
RIPK1 Q13546 3/20 0.40
ALDH1A1 P00352 1/20 0.40
GAA P10253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9877163 0.90 RAB9A (0.43) L3MBTL1CHRM2CHRM4CHRM5CHRM1
SCHEMBL4132243 0.80 RIPK1 (0.49) MEN1KMT2ATSHRRIPK1ALDH1A1
SCHEMBL11708369 0.77 KDM4E (0.66) L3MBTL1CHRM2CHRM4CHRM5CHRM1
SCHEMBL20646025 0.77 CHRM2 (0.47) L3MBTL1CHRM2CHRM4CHRM5CHRM1
SCHEMBL18366270 0.77 CHRM2 (0.47) L3MBTL1CHRM2CHRM4CHRM5CHRM1
SCHEMBL13225803 0.77 KDM4E (0.66) L3MBTL1CHRM2CHRM4CHRM5CHRM1
SCHEMBL3739324 0.76 HDAC6 (0.54) L3MBTL1CHRM2CHRM4CHRM5CHRM1
SCHEMBL5837860 0.75 L3MBTL1 (0.58) L3MBTL1CHRM2CHRM4CHRM5CHRM1
SCHEMBL2456072 0.74 CHRM2 (0.44) L3MBTL1CHRM2CHRM4CHRM5CHRM1
SCHEMBL24508712 0.74 CHRM2 (0.55) L3MBTL1CHRM2CHRM4CHRM5CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110023313-B Bicyclic amide compounds and methods of use thereof 豪夫迈·罗氏有限公司 2022-10-25 CN disclosed
CN-110072863-B RIP1 kinase inhibitors and methods of use 豪夫迈·罗氏有限公司 2022-08-30 CN disclosed
CN-110914271-A Bicyclic ketone compounds and methods of use thereof 豪夫迈·罗氏有限公司 2020-03-24 CN disclosed