SCHEMBL28414737

SCHEMBL28414737

Cc1ccc(C(C)(O)C#Cc2ccccc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.46
VCP P55072 1/20 0.45
MEN1 O00255 4/20 0.40
KMT2A Q03164 4/20 0.40
ALDH1A1 P00352 1/20 0.40
POLB P06746 1/20 0.40
TSHR P16473 2/20 0.39
NR1H2 P55055 2/20 0.38
APP P05067 1/20 0.38
RARB P10826 1/20 0.35
RARG P13631 1/20 0.35
CA12 O43570 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35
LMNA P02545 1/20 0.34
ALOX12 P18054 1/20 0.34
ACHE P22303 1/20 0.34
KIF11 P52732 1/20 0.34
ASIC3 Q9UHC3 1/20 0.33
CYP19A1 P11511 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19130510 1.00 MAPT (0.46) MAPTVCPMEN1KMT2AALDH1A1
SCHEMBL28408574 0.93 MAPT (0.42) MAPTVCPMEN1KMT2AALDH1A1
SCHEMBL523695 0.89 MAPT (0.51) MAPTKMT2AALDH1A1NR1H2APP
SCHEMBL28407155 0.84 KMT2A (0.47) MAPTMEN1KMT2AALDH1A1TSHR
SCHEMBL23064948 0.82 VCP (0.45) MAPTVCPMEN1KMT2AALDH1A1
SCHEMBL19148941 0.81 L3MBTL1 (0.47) MAPTMEN1KMT2AALDH1A1POLB
SCHEMBL19124263 0.81 L3MBTL1 (0.47) MAPTMEN1KMT2AALDH1A1POLB
SCHEMBL28604749 0.77 TSHR (0.43) MAPTMEN1ALDH1A1TSHRCA12
SCHEMBL4800627 0.77 MAPT (0.40) MAPTMEN1KMT2AALDH1A1TSHR
SCHEMBL23064944 0.76 ALDH1A1 (0.44) MAPTVCPMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108689893-B Propargyl sulfone compound and preparation method and application thereof 南京工业大学 2020-05-08 CN claimed
CN-108689893-B Propargyl sulfone compound and preparation method and application thereof 南京工业大学 2020-05-08 CN disclosed