SCHEMBL28421990

SCHEMBL28421990

CCCCNC(=O)c1nc2ccccc2nc1Sc1ccc(Br)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 4/20 0.46
TP53 P04637 2/20 0.44
HTT P42858 2/20 0.44
TSHR P16473 1/20 0.44
HPGD P15428 1/20 0.43
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA3 P07451 1/20 0.42
CA4 P22748 1/20 0.42
CA6 P23280 1/20 0.42
CA5A P35218 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42
CA13 Q8N1Q1 1/20 0.42
CA14 Q9ULX7 1/20 0.42
CA5B Q9Y2D0 1/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28416681 0.97 RXFP1 (0.43) RXFP1TP53HTTTSHRHPGD
SCHEMBL28416663 0.89 MEN1 (0.40) TP53HTTCA2CA4MEN1
SCHEMBL28419925 0.85 SMN1; SMN2 (0.49) TP53HPGDCA2ALDH1A1MAPT
SCHEMBL28796059 0.85 KMT2A (0.41) RXFP1TP53HTTMEN1KMT2A
SCHEMBL28426850 0.83 ALDH1A1 (0.43) RXFP1TP53HTTCA2MEN1
SCHEMBL28416682 0.81 L3MBTL1 (0.37) TP53HTTMEN1KMT2AMAPT
SCHEMBL28421991 0.78 KMT2A (0.37) TP53HTTMEN1KMT2AMAPT
SCHEMBL28427552 0.76 TARBP2 (0.46) HTTMEN1KMT2APOLBALDH1A1
SCHEMBL29889909 0.75 MEN1 (0.46) HTTMEN1KMT2AALDH1A1MAPT
SCHEMBL28945793 0.73 KDM4E (0.44) RXFP1TP53HTTCA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110981819-A Quinoxaline signal channel inhibitor and preparation method and application thereof 广西师范大学 2020-04-10 CN disclosed