SCHEMBL28429223

SCHEMBL28429223

O=C1CN(C(=O)OCc2ccccc2)CCN1CC1CCCC1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP19 O94966 1/20 0.55
SMN1; SMN2 Q16637 3/20 0.52
NPC1 O15118 2/20 0.52
RAB9A P51151 2/20 0.52
CYP2C19 P33261 1/20 0.50
P2RX7 Q99572 2/20 0.48
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
TMEM97 Q5BJF2 5/20 0.46
SIGMAR1 Q99720 5/20 0.46
HTR1A P08908 2/20 0.46
HRH2 P25021 2/20 0.46
HRH1 P35367 2/20 0.46
HRH3 Q9Y5N1 2/20 0.46
CHRM4 P08173 1/20 0.46
CHRM5 P08912 1/20 0.46
ADRA2A P08913 1/20 0.46
ADRA2B P18089 1/20 0.46
ADRA1D P25100 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28437662 0.99 USP19 (0.56) USP19SMN1; SMN2NPC1RAB9ACYP2C19
SCHEMBL25251265 0.90 SMN1; SMN2 (0.49) USP19SMN1; SMN2NPC1RAB9ACYP2C19
SCHEMBL7657420 0.85 SMN1; SMN2 (0.50) USP19SMN1; SMN2NPC1RAB9ACYP2C19
SCHEMBL4385886 0.85 SMN1; SMN2 (0.50) USP19SMN1; SMN2NPC1RAB9ACYP2C19
SCHEMBL3902852 0.83 SMN1; SMN2 (0.56) USP19SMN1; SMN2NPC1RAB9ACYP2C19
SCHEMBL20339027 0.82 PARP1 (0.46) USP19SMN1; SMN2NPC1RAB9ACYP2C19
SCHEMBL8386105 0.82 KMT2A (0.52) USP19SMN1; SMN2NPC1RAB9ACYP2C19
SCHEMBL30288951 0.81 DRD2 (0.52) USP19SMN1; SMN2NPC1RAB9AMEN1
SCHEMBL28435744 0.81 SMN1; SMN2 (0.54) USP19SMN1; SMN2NPC1RAB9ACYP2C19
SCHEMBL25426557 0.81 SMN1; SMN2 (0.45) USP19SMN1; SMN2NPC1RAB9ACYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107098886-B Prazinone-containing quinazolinone PARP-1/2 inhibitor and preparation method, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2020-07-14 CN disclosed