SCHEMBL28434865

SCHEMBL28434865

C[Si](C)(C)CCOCn1cnc(C=O)n1

nearest known ligand 0.33

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 1/20 0.31
NPC1 O15118 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24306335 0.79 DGAT1 (0.35) DGAT1
SCHEMBL951764 0.78 DGAT1 (0.37) DGAT1
SCHEMBL1811528 0.78 ALOX5AP (0.33) DGAT1NPC1
SCHEMBL23939802 0.78 DGAT1 (0.32) DGAT1NPC1
SCHEMBL29961918 0.78 DGAT1 (0.32) DGAT1
SCHEMBL949085 0.77 ALDH1A1 (0.43) DGAT1
SCHEMBL20272451 0.77 DGAT1 (0.30) DGAT1
SCHEMBL953734 0.76 DGAT1 (0.36) DGAT1
SCHEMBL16387217 0.76 NPC1 (0.36) DGAT1NPC1
SCHEMBL18863096 0.76 SMN1; SMN2 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111556871-B 1H-pyrazolo [4,3-b ] pyridines as PDE1 inhibitors H.隆德贝克有限公司 2023-07-07 CN disclosed
CN-111465410-B Combination therapy comprising administration of 1H-pyrazolo [4,3-B ] pyridine H.隆德贝克有限公司 2022-10-25 CN disclosed
CN-111526890-B Combination therapy comprising administration of 1H-pyrazolo [4,3-B ] pyridine H.隆德贝克有限公司 2022-10-14 CN disclosed
CN-109311872-B 1H-pyrazolo [4,3-b ] pyridines as PDE1 inhibitors H.隆德贝克有限公司 2021-08-20 CN disclosed
CN-111556871-A 1H-pyrazolo [4,3-b ] pyridines as PDE1 inhibitors H.隆德贝克有限公司 2020-08-18 CN disclosed
CN-111526890-A Combination therapy comprising administration of 1H-pyrazolo [4,3-B ] pyridine H.隆德贝克有限公司 2020-08-11 CN disclosed
CN-111465410-A Combination therapy comprising administration of 1H-pyrazolo [4,3-B ] pyridine H.隆德贝克有限公司 2020-07-28 CN disclosed