SCHEMBL951764

SCHEMBL951764

C[Si](C)(C)CCOCn1cnc(Br)n1

nearest known ligand 0.37

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 3/20 0.37
HDAC1 Q13547 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL953734 0.98 DGAT1 (0.36) DGAT1HDAC1HDAC6
SCHEMBL953732 0.97 DGAT1 (0.36) DGAT1HDAC1HDAC6
SCHEMBL24306335 0.81 DGAT1 (0.35) DGAT1
SCHEMBL1811528 0.80 ALOX5AP (0.33) DGAT1
SCHEMBL23939802 0.80 DGAT1 (0.32) DGAT1
SCHEMBL29961918 0.80 DGAT1 (0.32) DGAT1
SCHEMBL3508159 0.79 DGAT1 (0.40) DGAT1HDAC1HDAC6
SCHEMBL28434865 0.78 DGAT1 (0.31) DGAT1
SCHEMBL16847388 0.78 DGAT1 (0.31) DGAT1
SCHEMBL19284804 0.78 DGAT1 (0.31) DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 47 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4703357-A1 TRIAZOLYL-CONTAINING COMPOUNDS Chia Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2026-03-04 EP disclosed
US-12552767-B2 3-heteroaryl pyrrolidine and piperidine orexin receptor agonists MERCK SHARP & DOHME LLC (US) 2026-02-17 US disclosed
EP-4587435-A1 MODIFIED PROTEINS AND PROTEIN BINDERS AND DEGRADERS Cullgen (Shanghai), Inc. (CN) 2025-07-23 EP disclosed
US-20250215030-A1 STAT MODULATORS AND USES THEREOF RECLUDIX PHARMA, INC. 2025-07-03 US disclosed
WO-2025096495-A1 ARYL FLUOROSULFATE-BASED INHIBITORS AS NOVEL ANTITUBERCULAR AGENTS THE SCRIPPS RESEARCH INSTITUTE (US) 2025-05-08 WO disclosed
US-20250115597-A1 TYK2 INHIBITORS AND COMPOSITIONS AND METHODS THEREOF LYNK PHARMACEUTICALS CO LTD (CN) 2025-04-10 US disclosed
US-20250091994-A1 RAS/RAF BINDING INHIBITOR COMPOUND NATIONAL UNIVERSITY CORPORATION KOBE UNIVERSITY (JP) 2025-03-20 US disclosed
EP-4499656-A1 STAT MODULATORS AND USES THEREOF Recludix Pharma, Inc. (US) 2025-02-05 EP disclosed
US-20250002472-A1 PYRIDYL-CONTAINING COMPOUND CHIA TAI TIANQING PHARMACEUTICAL GROUP CO., LTD. (CN) 2025-01-02 US disclosed
CN-119183453-A STAT modulators and uses thereof 瑞克鲁迪克斯制药股份有限公司 2024-12-24 CN disclosed
US-20170137430-A1 Nuclear Transport Modulators And Uses Thereof KARYOPHARM THERAPEUTICS INC (US) 2017-05-18 US disclosed
US-9428490-B2 Nuclear transport modulators and uses thereof Karyopharm Therapeutics Inc. (US) 2016-08-30 US disclosed
US-9428490-B2 Nuclear transport modulators and uses thereof Karyopharm Therapeutics Inc. (US) 2016-08-30 US disclosed
US-9428490-B2 Nuclear transport modulators and uses thereof Karyopharm Therapeutics Inc. (US) 2016-08-30 US disclosed
EP-2736883-A1 NUCLEAR TRANSPORT MODULATORS AND USES THEREOF Karyopharm Therapeutics, Inc. (US) 2014-06-04 EP disclosed
WO-2013019561-A1 NUCLEAR TRANSPORT MODULATORS AND USES THEREOF KARYOPHARM THERAPEUTICS, INC. (US) 2013-02-07 WO disclosed
WO-2013019561-A1 NUCLEAR TRANSPORT MODULATORS AND USES THEREOF KARYOPHARM THERAPEUTICS, INC. (US) 2013-02-07 WO disclosed
US-20120128630-A1 1-(6 MEMBERS AZO-HETEROCYCLIC)-PYRROLIN-2-ONE COMPOUNDS AS INHIBITORS OF HEPATITIS C NS5B POLYMERASE, THE PHARAMACEUTICAL COMPOSITION THEREOF AND THEIR THERAPEUTIC USE VIVALIS (FR) 2012-05-24 US disclosed
EP-2451800-A1 1-(6 MEMBERS AZO-HETEROCYCLIC)-PYRROLIN-2-ONE COMPOUNDS AS INHIBITORS OF HEPATITIS C NS5B POLYMERASE, THE PHARMACEUTICAL COMPOSITION THEREOF AND THEIR THERAPEUTIC USE Vivalis (FR) 2012-05-16 EP disclosed
WO-2011004017-A1 1-(6 MEMBERS AZO-HETEROCYCLIC)-PYRROLIN-2-ONE COMPOUNDS AS INHIBITORS OF HEPATITIS C NS5B POLYMERASE, THE PHARMACEUTICAL COMPOSITION THEREOF AND THEIR THERAPEUTIC USE VIVALIS (FR) 2011-01-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250091994-A1 RAS/RAF BINDING INHIBITOR COMPOUND BRAF, RAF1, NRAS DGAT1 3556/4885HDAC1 1396/4885HDAC6 2237/4885
US-20250215030-A1 STAT MODULATORS AND USES THEREOF STAT6, STAT3, STAT5A DGAT1 3167/4885HDAC1 227/4885HDAC6 110/4885
US-20120128630-A1 1-(6 MEMBERS AZO-HETEROCYCLIC)-PYRROLIN-2-ONE COMPOUNDS AS INHIBITORS OF HEPATITIS C NS5B POLYMERASE, THE PHARAMACEUTICAL COMPOSITION THEREOF AND THEIR THERAPEUTIC USE NAT1, POLM, PYGL DGAT1 2530/4885HDAC1 454/4885HDAC6 433/4885
US-12552767-B2 3-heteroaryl pyrrolidine and piperidine orexin receptor agonists HCRTR2, HCRTR1, NPY1R DGAT1 3006/4885HDAC1 582/4885HDAC6 742/4885
US-20170137430-A1 Nuclear Transport Modulators And Uses Thereof XPO1, XPO5, XPOT DGAT1 3640/4885HDAC1 199/4885HDAC6 204/4885
US-20250002472-A1 PYRIDYL-CONTAINING COMPOUND DPYD, TYMP, WEE1 DGAT1 4767/4885HDAC1 1048/4885HDAC6 2326/4885
US-20250115597-A1 TYK2 INHIBITORS AND COMPOSITIONS AND METHODS THEREOF TYK2, JAK2, JAK1 DGAT1 3938/4885HDAC1 1415/4885HDAC6 706/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.