SCHEMBL28436348

SCHEMBL28436348

COc1c(OC)c2cccc3c(C#N)c(C#N)c4cccc1c4c32

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.43
ALDH1A1 P00352 4/20 0.43
MAPK1 P28482 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
IMPDH2 P12268 1/20 0.39
IMPDH1 P20839 1/20 0.39
MAPT P10636 4/20 0.38
MEN1 O00255 2/20 0.38
GAA P10253 2/20 0.38
KMT2A Q03164 2/20 0.38
CACNA1B Q00975 1/20 0.38
APBA1 Q02410 1/20 0.38
SQOR Q9Y6N5 3/20 0.37
POLB P06746 2/20 0.35
MAOA P21397 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
ADORA2A P29274 2/20 0.34
ADORA1 P30542 2/20 0.34
AKR1B1 P15121 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20718126 0.82 ALDH1A1 (0.50) KDM4EALDH1A1IMPDH2IMPDH1MAPT
SCHEMBL4958710 0.77 KDM4E (0.61) KDM4EALDH1A1MAPK1SMN1; SMN2IMPDH2
SCHEMBL28415690 0.77 ALDH1A1 (0.41) KDM4EALDH1A1MAPK1MAPTMEN1
SCHEMBL31171419 0.77 KDM4E (0.61) KDM4EALDH1A1MAPK1SMN1; SMN2IMPDH2
SCHEMBL28864503 0.72 ALDH1A1 (0.48) KDM4EALDH1A1MAPK1SMN1; SMN2MAPT
SCHEMBL28313759 0.70 KDM4E (0.64) KDM4EALDH1A1MAPK1SMN1; SMN2IMPDH2
SCHEMBL28858809 0.68 ALDH1A1 (0.43) KDM4EALDH1A1MAPK1SMN1; SMN2MAPT
SCHEMBL6736896 0.67 POLB (0.47) KDM4EALDH1A1MAPK1SMN1; SMN2IMPDH2
SCHEMBL4739158 0.67 RAB9A (0.59) KDM4EALDH1A1MAPK1SMN1; SMN2IMPDH2
SCHEMBL25017593 0.67 NQO1 (0.50) KDM4EALDH1A1MAPK1MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108658993-B Pyreneimide derivative and synthesis method and application thereof 兰州大学 2020-07-10 CN disclosed