SCHEMBL28439261

SCHEMBL28439261

CC(C)c1cc(-c2ccccn2)c(O)c(-c2ccccn2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.43
LMNA P02545 3/20 0.43
CCR1 P32246 2/20 0.43
CCR5 P51681 2/20 0.43
CCR8 P51685 2/20 0.43
CYP1A2 P05177 1/20 0.43
POLB P06746 1/20 0.43
METAP1 P53582 1/20 0.43
BLM P54132 1/20 0.43
HIF1A Q16665 1/20 0.43
DOHH Q9BU89 1/20 0.43
P4HTM Q9NXG6 1/20 0.43
TDP1 Q9NUW8 2/20 0.42
KDM1A O60341 3/20 0.42
TGFBR1 P36897 1/20 0.42
HTT P42858 3/20 0.41
MAOA P21397 1/20 0.41
BRD4 O60885 2/20 0.40
BRD2 P25440 1/20 0.40
BRD3 Q15059 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10299991 0.80 KDM4E (0.48) KDM4ELMNACCR1CCR5CCR8
SCHEMBL20232781 0.78 TGFBR1 (0.39) KDM4ELMNACCR1CCR5CCR8
SCHEMBL11996115 0.77 CCR1 (0.58) KDM4ELMNACCR1CCR5CCR8
SCHEMBL1102459 0.77 KDM4E (0.48) KDM4ELMNACCR1CCR5CCR8
SCHEMBL14864003 0.76 KDM4E (0.43) KDM4ELMNACCR1CCR5CCR8
SCHEMBL14864032 0.76 METAP2 (0.44) KDM4ELMNACCR1CCR5CCR8
SCHEMBL2734583 0.75 KDM4E (0.56) KDM4ELMNACCR1CCR5CCR8
Dipyridyl SCHEMBL28441671 0.75 KDM4E (0.52) KDM4ELMNACCR1CCR5CCR8
SCHEMBL28218416 0.75 KDM4E (0.46) KDM4ELMNACCR1CCR5CCR8
SCHEMBL4565295 0.75 HSP90AA1 (0.49) KDM4ELMNACCR1CCR5CCR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111454198-A Compound based on dipyridyl phenol/thiophenol and preparation method and application thereof 复旦大学 2020-07-28 CN disclosed