SCHEMBL28440477

SCHEMBL28440477

COc1cccc2c1C(=O)c1c(OC)cc(CN3CCN(c4ccccn4)CC3)cc1C2=O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.56
KDM4E B2RXH2 5/20 0.56
TSHR P16473 3/20 0.56
LMNA P02545 3/20 0.56
HTT P42858 2/20 0.56
MAPK1 P28482 1/20 0.56
DRD4 P21917 3/20 0.50
DRD3 P35462 3/20 0.50
DRD2 P14416 2/20 0.50
SIGMAR1 Q99720 2/20 0.49
HTR2A P28223 1/20 0.48
HPGD P15428 3/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
ALOX12 P18054 1/20 0.48
HSD17B10 Q99714 2/20 0.47
HTR1A P08908 3/20 0.47
ADRA1D P25100 1/20 0.46
ADRA1A P35348 1/20 0.46
ADRA1B P35368 1/20 0.46
MAPT P10636 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28446165 0.89 DRD2 (0.60) ALDH1A1KDM4EMAPK1DRD4DRD3
SCHEMBL28897363 0.85 MAPT (0.52) ALDH1A1SIGMAR1MAPT
SCHEMBL28439934 0.82 NPC1 (0.46) LMNAMAPK1HSD17B10MAPT
SCHEMBL28446805 0.82 ACHE (0.46) LMNADRD4DRD3DRD2MAPT
SCHEMBL28440012 0.82 ALDH1A1 (0.62) ALDH1A1KDM4ETSHRLMNAMAPK1
SCHEMBL28897885 0.81 GAA (0.51)
SCHEMBL28446037 0.81 KDM4E (0.52) ALDH1A1KDM4ELMNAHTTMAPK1
SCHEMBL28444429 0.80 TDP1 (0.46) ALDH1A1KDM4ELMNAMAPT
SCHEMBL28450388 0.79 HTR7 (0.45) HTR2AHTR1AMAPT
SCHEMBL28447509 0.79 PDE4B (0.50) ALDH1A1LMNAHTTDRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111592479-B Aloe-emodin nitrogen heterocyclic derivative and preparation method and application thereof 四川大学华西医院 2021-10-19 CN disclosed
CN-111592479-A Aloe-emodin nitrogen heterocyclic derivative and preparation method and application thereof 四川大学华西医院 2020-08-28 CN disclosed