SCHEMBL28443306

SCHEMBL28443306

COC(=O)C1=C(C)NC(C)=C(C(=O)OCCC#N)C1c1ccc(Cl)cc1Cl

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 4/20 0.53
KDM4E B2RXH2 4/20 0.53
ALDH1A1 P00352 4/20 0.53
HSD17B10 Q99714 3/20 0.53
CYP3A4 P08684 3/20 0.53
CYP2C19 P33261 3/20 0.53
ABCB11 O95342 3/20 0.53
TBXA2R P21731 3/20 0.53
ADRA1A P35348 3/20 0.53
SLC6A3 Q01959 3/20 0.53
ADORA3 P0DMS8 3/20 0.53
MEN1 O00255 2/20 0.53
CYP1A2 P05177 2/20 0.53
KMT2A Q03164 2/20 0.53
HIF1A Q16665 2/20 0.53
MAPT P10636 2/20 0.53
ABCB1 P08183 2/20 0.53
ADRB3 P13945 2/20 0.53
OPRK1 P41145 2/20 0.53
SCN5A Q14524 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8518663 0.87 ABCB11 (0.61) CYP2C9KDM4EALDH1A1HSD17B10CYP3A4
SCHEMBL820500 0.85 CYP2C9 (0.74) CYP2C9KDM4EALDH1A1HSD17B10CYP3A4
SCHEMBL29808878 0.85 CYP2C9 (0.74) CYP2C9KDM4EALDH1A1HSD17B10CYP3A4
SCHEMBL29676455 0.85 ALDH1A1 (0.59) CYP2C9KDM4EALDH1A1HSD17B10CYP3A4
SCHEMBL3028387 0.85 ALDH1A1 (0.59) CYP2C9KDM4EALDH1A1HSD17B10CYP3A4
SCHEMBL28441003 0.82 CACNA1F (0.53) CYP2C9KDM4EALDH1A1HSD17B10CYP3A4
SCHEMBL28438034 0.81 ALDH1A1 (0.55) CYP2C9KDM4EALDH1A1HSD17B10CYP3A4
SCHEMBL3016247 0.81 MAPK1 (0.70) CYP2C9KDM4EALDH1A1HSD17B10CYP3A4
SCHEMBL5855031 0.81 CACNA1B (0.63) CACNA1CCACNA1FCACNA1DCACNA1SABCC1
SCHEMBL11105563 0.79 NR1I2 (0.56) CYP2C9KDM4EALDH1A1HSD17B10CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111423362-A Preparation method of two high-purity clevidipine butyrate impurities 山东省药学科学院 2020-07-17 CN disclosed