SCHEMBL8518663

SCHEMBL8518663

COC(=O)C1=C(C)NC(C)=C(C(=O)OCCC#N)C1c1ccccc1Cl

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB11 O95342 5/20 0.61
ADORA3 P0DMS8 5/20 0.61
CYP2C9 P11712 4/20 0.61
ADRA1A P35348 4/20 0.61
CYP3A4 P08684 4/20 0.61
CYP1A2 P05177 4/20 0.61
SCN5A Q14524 4/20 0.61
TBXA2R P21731 3/20 0.61
SLC6A3 Q01959 3/20 0.61
KDM4E B2RXH2 3/20 0.61
CYP2C19 P33261 3/20 0.61
KMT2A Q03164 3/20 0.61
HIF1A Q16665 3/20 0.61
HSD17B10 Q99714 3/20 0.61
ABCB1 P08183 3/20 0.61
NR1I2 O75469 3/20 0.61
LMNA P02545 3/20 0.61
SCN1A P35498 3/20 0.61
SCN2A Q99250 3/20 0.61
SCN3A Q9NY46 3/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL820500 0.92 CYP2C9 (0.74) ABCB11ADORA3CYP2C9ADRA1ACYP3A4
SCHEMBL29808878 0.92 CYP2C9 (0.74) ABCB11ADORA3CYP2C9ADRA1ACYP3A4
SCHEMBL8297064 0.88 ALDH1A1 (0.53) ABCB11ADORA3CYP2C9ADRA1ACYP3A4
SCHEMBL28443306 0.87 CYP2C9 (0.53) ABCB11ADORA3CYP2C9ADRA1ACYP3A4
SCHEMBL11105563 0.87 NR1I2 (0.56) ABCB11ADORA3CYP2C9ADRA1ACYP3A4
SCHEMBL9485304 0.86 ABCB11 (0.72) ABCB11ADORA3CYP2C9ADRA1ACYP3A4
SCHEMBL27421079 0.86 CYP2C9 (0.69) ABCB11ADORA3CYP2C9ADRA1ACYP3A4
SCHEMBL8298008 0.86 TBXA2R (0.47) ABCB11ADORA3CYP2C9ADRA1ACYP3A4
SCHEMBL10822224 0.85 KDM4E (0.47) ABCB11ADORA3CYP2C9ADRA1ACYP3A4
SCHEMBL3031020 0.85 ADORA3 (0.82) ABCB11ADORA3CYP2C9ADRA1ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012065527-A1 COMPOUDS AND USES AS L-TYPE CALCIUM CHANNEL BLOCKER AND/OR ACETYLCHOLINESTERASE INHIBITOR THEREOF 江苏先声药物研究有限公司 (CN) 2012-05-24 WO disclosed