SCHEMBL28445883

SCHEMBL28445883

OC1N=Cc2ccccc21

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
HTR2A P28223 1/20 0.31
CYP2D6 P10635 1/20 0.31
MEN1 O00255 1/20 0.30
GAA P10253 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9545204 0.83 CYP2D6 (0.34) HTR2ACYP2D6MEN1KMT2A
SCHEMBL23513879 0.73 EDNRA (0.32)
SCHEMBL6045293 0.71 HTR2A (0.35) HTR2AMEN1GAAKMT2A
SCHEMBL8527375 0.71 HTR5A (0.33) HTR2A
SCHEMBL29354632 0.70 KDM1A (0.37) HTR2AMEN1GAAKMT2A
Hydrochloric Acid SCHEMBL7724483 0.70 KDM1A (0.36) HTR2A
SCHEMBL3750452 0.69 ATM (0.43) HTR2AMEN1GAAKMT2A
SCHEMBL9298612 0.67 POLB (0.34)
SCHEMBL19696034 0.67 KDM1A (0.31)
SCHEMBL24596781 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111499580-A Substituted diaminocarboxamides and diaminocarbonitrile pyrimidines, compositions thereof, and methods of treatment therewith 西格诺药品有限公司 2020-08-07 CN disclosed
CN-111471021-A Substituted diaminocarboxamides and diaminocarbonitrile pyrimidines, compositions thereof, and methods of treatment therewith 西格诺药品有限公司 2020-07-31 CN disclosed