SCHEMBL9298612

SCHEMBL9298612

O=C(O)OC1N=Cc2ccccc21

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.34
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
EDNRA P25101 2/20 0.32
HDAC4 P56524 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.31
HTT P42858 1/20 0.30
EDNRB P24530 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27546882 0.81 HCAR2 (0.32) POLBKDM4E
SCHEMBL3750452 0.68 ATM (0.43) POLBALDH1A1HDAC4
SCHEMBL28445883 0.67 MAOA (0.33)
SCHEMBL30931450 0.67 POLB (0.38) POLBKDM4EALDH1A1EDNRAHDAC4
SCHEMBL18921545 0.64 CYP2D6 (0.41) POLBKDM4EALDH1A1EDNRAEDNRB
SCHEMBL23513879 0.64 EDNRA (0.32) ALDH1A1EDNRA
SCHEMBL4607072 0.64 SLC6A2 (0.40) POLBEDNRAPTGDR2
SCHEMBL7596802 0.64 POLB (0.52) POLBEDNRAHDAC4EDNRB
SCHEMBL28044427 0.63 HTR2A (0.31)
SCHEMBL27300866 0.63

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0629211-A1 4-OXO-2 THIOXOIMIDAZOLIDINE DERIVATES AS INHIBITORS OF BLOOD PLATELET AGGREGATION HOECHST AKTIENGESELLSCHAFT (DE) 1994-12-21 EP disclosed
WO-1993018057-A1 4-OXO-2 THIOXOIMIDAZOLIDINE DERIVATES AS INHIBITORS OF BLOOD PLATELET AGGREGATION CASSELLA AKTIENGESELLSCHAFT (DE) 1993-09-16 WO disclosed
EP-0115345-A1 Process for the resolution of racemic optically active bicyclic imino-alpha-carboxylic acid esters and use of the compounds obtainable in this way for the synthesis of carboxyalkyl dipeptides HOECHST AKTIENGESELLSCHAFT (DE) 1984-08-08 EP disclosed