SCHEMBL28447402

SCHEMBL28447402

O=C(O)C1(c2ncc(-c3ccccc3Cl)cn2)C=CC=CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 3/20 0.39
EGLN3 Q9H6Z9 2/20 0.37
MAP4K4 O95819 1/20 0.36
ABL1 P00519 2/20 0.36
NPY5R Q15761 1/20 0.36
CNR2 P34972 1/20 0.36
DEGS1 O15121 1/20 0.36
CYP2A6 P11509 1/20 0.35
USP7 Q93009 1/20 0.34
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP11B1 P15538 1/20 0.33
VEGFA P15692 1/20 0.33
FLT1 P17948 1/20 0.33
CNR1 P21554 1/20 0.33
PDE4B Q07343 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
ATM Q13315 1/20 0.32
DHODH Q02127 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzene SCHEMBL28354853 0.69 HDAC4 (0.41)
SCHEMBL4451679 0.69 HDAC4 (0.41)
SCHEMBL8626071 0.68 L3MBTL1 (0.36) CNR2KDM4EALDH1A1
SCHEMBL11477196 0.67 USP7 (0.53) EGLN1EGLN3MAP4K4CNR2DEGS1
SCHEMBL27731834 0.66 AKR1C1 (0.37) KDM4EALDH1A1NPC1
SCHEMBL8424787 0.64 TSHR (0.38) ALDH1A1
SCHEMBL4780143 0.64 EGLN1 (0.56) EGLN1EGLN3MAP4K4CNR2DEGS1
SCHEMBL29120630 0.64 HDAC4 (0.39) CYP11B1
SCHEMBL28755670 0.64 HDAC4 (0.39) CYP11B1
SCHEMBL10899864 0.63 CYP2A6 (0.56) EGLN1EGLN3MAP4K4ABL1NPY5R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107074812-B Substituted pyrimidine compounds 格吕伦塔尔有限公司 2020-08-21 CN disclosed