SCHEMBL28447449

SCHEMBL28447449

O=C(O)c1ccc2c(c1)N(CCBr)CC2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
MAPT P10636 2/20 0.46
KDM4E B2RXH2 1/20 0.46
POLB P06746 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
ALDH1A1 P00352 3/20 0.42
LMNA P02545 2/20 0.41
PMP22 Q01453 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
GFER P55789 1/20 0.41
ACHE P22303 1/20 0.41
KDM4C Q9H3R0 2/20 0.40
CHRM2 P08172 1/20 0.40
CHRM3 P20309 1/20 0.40
KDM4A O75164 1/20 0.40
KDM2B Q8NHM5 1/20 0.40
NPC1 O15118 1/20 0.40
NR4A1 P22736 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7213441 0.83 XIAP (0.47) MEN1KMT2AKDM4EPOLBALDH1A1
SCHEMBL3349545 0.83 ACHE (0.47) MEN1KMT2AMAPTKDM4EPOLB
SCHEMBL5404613 0.82 ACHE (0.46) MEN1KMT2AMAPTKDM4EPOLB
SCHEMBL6177893 0.78 ACHE (0.63) MAPTKDM4EALDH1A1ACHESLC22A12
SCHEMBL12193492 0.76 ALDH1A1 (0.49) KDM4EALDH1A1LMNAACHEMYC
SCHEMBL3350583 0.76 ALDH1A1 (0.48) MEN1KMT2AMAPTKDM4EL3MBTL1
SCHEMBL20178669 0.75 ACHE (0.53) MEN1KMT2AMAPTKDM4EL3MBTL1
SCHEMBL11977166 0.74 SLC22A12 (0.70) MAPTALDH1A1ACHESLC22A12MYC
SCHEMBL12359557 0.74 ACHE (0.41) MEN1KMT2AMAPTKDM4EPOLB
SCHEMBL4929256 0.73 ALDH1A1 (0.57) MEN1KMT2AMAPTKDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107074816-B Heterocyclic derivative, preparation method and medical application thereof 四川海思科制药有限公司 2020-07-17 CN disclosed