SCHEMBL28447724

SCHEMBL28447724

CC(C)(C)OC(=O)N1CCN(Cc2ccccc2N2CCCC2)CC1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 8/20 0.68
ABHD6 Q9BV23 8/20 0.68
PLA2G7 Q13093 6/20 0.68
TRPV1 Q8NER1 2/20 0.53
CHRM2 P08172 1/20 0.51
CHRM4 P08173 1/20 0.51
CHRM1 P11229 1/20 0.51
CHRM3 P20309 1/20 0.51
FAAH O00519 1/20 0.51
CYP2D6 P10635 1/20 0.49
ALDH1A1 P00352 2/20 0.49
KDM4E B2RXH2 1/20 0.49
POLB P06746 1/20 0.49
VEGFA P15692 1/20 0.48
EGLN1 Q9GZT9 1/20 0.48
GPR119 Q8TDV5 1/20 0.46
CKS1B P61024 1/20 0.45
SKP1 P63208 1/20 0.45
SKP2 Q13309 1/20 0.45
MEN1 O00255 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30141417 1.00 MGLL (0.68) MGLLABHD6PLA2G7TRPV1CHRM2
SCHEMBL5335100 0.95 PLA2G7 (0.61) MGLLABHD6PLA2G7TRPV1CHRM2
SCHEMBL5335298 0.94 MGLL (0.60) MGLLABHD6PLA2G7TRPV1CHRM2
SCHEMBL15264216 0.89 MGLL (0.55) MGLLABHD6PLA2G7TRPV1CHRM2
SCHEMBL15264833 0.88 MGLL (0.54) MGLLABHD6PLA2G7TRPV1CHRM2
SCHEMBL5336442 0.87 MGLL (0.53) MGLLABHD6PLA2G7CHRM2CHRM4
SCHEMBL28630470 0.86 PLA2G7 (0.53) MGLLABHD6PLA2G7TRPV1CHRM2
SCHEMBL7986047 0.85 CKS1B (0.57) MGLLABHD6PLA2G7CHRM2CHRM4
SCHEMBL15265005 0.84 MGLL (0.50) MGLLABHD6PLA2G7TRPV1CHRM2
SCHEMBL16744505 0.84 MGLL (0.54) MGLLABHD6PLA2G7TRPV1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111454233-B 4- (2- (pyrrolidine/piperidine-1-yl) benzyl) -piperazinylurea TRPV1 antagonist and preparation and application thereof 河南大学 2023-01-24 CN disclosed
CN-111454233-A 4- (2- (pyrrolidine/piperidine-1-yl) benzyl) -piperazinylurea TRPV1 antagonist and preparation and application thereof 河南大学 2020-07-28 CN disclosed