SCHEMBL28630470

SCHEMBL28630470

CC(C)(C)OC(=O)N1CCN(Cc2ccccc2N2CCC(c3ccccc3)CC2)CC1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PLA2G7 Q13093 1/20 0.53
MGLL Q99685 1/20 0.53
ABHD6 Q9BV23 1/20 0.53
GPR119 Q8TDV5 2/20 0.52
NAMPT P43490 1/20 0.49
FAAH O00519 2/20 0.49
TRPV1 Q8NER1 2/20 0.49
CHRM4 P08173 2/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
TP53 P04637 3/20 0.47
THRB P10828 1/20 0.47
MAPT P10636 1/20 0.47
CHRM2 P08172 1/20 0.46
CHRM1 P11229 1/20 0.46
CHRM3 P20309 1/20 0.46
KDM4E B2RXH2 1/20 0.45
PKM P14618 1/20 0.45
PIK3CD O00329 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30632156 0.88 MGLL (0.56) PLA2G7MGLLABHD6FAAH
SCHEMBL28614777 0.88 MGLL (0.56) PLA2G7MGLLABHD6FAAH
SCHEMBL28447724 0.86 MGLL (0.68) PLA2G7MGLLABHD6GPR119FAAH
SCHEMBL30141417 0.86 MGLL (0.68) PLA2G7MGLLABHD6GPR119FAAH
SCHEMBL5335100 0.84 PLA2G7 (0.61) PLA2G7MGLLABHD6GPR119FAAH
SCHEMBL5335298 0.83 MGLL (0.60) PLA2G7MGLLABHD6GPR119FAAH
SCHEMBL3843148 0.82 NAMPT (0.66) GPR119NAMPTMEN1KMT2ATP53
SCHEMBL6132848 0.82 GPR119 (0.69) GPR119NAMPTTP53MAPT
SCHEMBL28613846 0.81 OPRM1 (0.55) PLA2G7MGLLABHD6MEN1KMT2A
SCHEMBL5336442 0.81 MGLL (0.53) PLA2G7MGLLABHD6GPR119NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113292485-B Benzyl piperazine urea TRPV1 antagonizing and MOR agonizing double-target medicine and its prepn and application 河南大学 2023-10-27 CN disclosed
CN-113292485-A Benzylpiperazine urea TRPV1 antagonistic and MOR agonistic double-target-point medicine, preparation method and application 河南大学 2021-08-24 CN disclosed