SCHEMBL28450201

SCHEMBL28450201

COc1cccc(F)c1-c1ccc2nn(C3CCN(C(=O)OC(C)(C)C)CC3)cc2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 2/20 0.44
IRAK4 Q9NWZ3 9/20 0.43
ALDH1A1 P00352 2/20 0.43
LMNA P02545 1/20 0.43
DNMT3A Q9Y6K1 1/20 0.42
CACNB4 O00305 1/20 0.42
CACNA1A O00555 1/20 0.42
CACNA1G O43497 1/20 0.42
CACNG3 O60359 1/20 0.42
CACNA1F O60840 1/20 0.42
CACNA1H O95180 1/20 0.42
CACNB3 P54284 1/20 0.42
CACNA2D1 P54289 1/20 0.42
CACNG7 P62955 1/20 0.42
CACNA1B Q00975 1/20 0.42
CACNA1D Q01668 1/20 0.42
CACNB1 Q02641 1/20 0.42
CACNG1 Q06432 1/20 0.42
CACNB2 Q08289 1/20 0.42
CACNA1S Q13698 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28452368 0.93 IRAK4 (0.43) GPR119IRAK4ALDH1A1LMNADNMT3A
SCHEMBL28460224 0.91 CACNB4 (0.41) IRAK4ALDH1A1LMNADNMT3ACACNB4
SCHEMBL28455484 0.90 APLNR (0.42) ALDH1A1LMNAFGFR3KDR
SCHEMBL28449757 0.85 EGFR (0.44) IRAK4FGFR4
SCHEMBL28898155 0.85 JAK2 (0.45) GPR119ALDH1A1JAK2JAK3PTK2
SCHEMBL28898962 0.84 CACNB4 (0.41) IRAK4ALDH1A1LMNADNMT3ACACNB4
SCHEMBL28456326 0.84 APLNR (0.42) ALDH1A1LMNAFGFR3KDR
SCHEMBL28457706 0.82 GPR119 (0.42) GPR119ALDH1A1LMNADNMT3ACACNB4
SCHEMBL25204156 0.79 GPR119 (0.44) GPR119TTKJAK2JAK3PTK2
SCHEMBL28450193 0.78 BTK (0.42) FGFR1FGFR2FGFR4FGFR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111662232-B Small molecule compound with 2H-indazole structure and synthesis and application thereof 中国科学院上海药物研究所 2022-08-02 CN disclosed
CN-111662232-A Small molecule compound with 2H-indazole structure and synthesis and application thereof 中国科学院上海药物研究所 2020-09-15 CN disclosed