SCHEMBL28455484

SCHEMBL28455484

COc1cccc(F)c1-c1ccc2nn(C3CCCN(C(=O)OC(C)(C)C)C3)cc2c1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
APLNR P35414 1/20 0.42
PIK3CD O00329 2/20 0.40
PIK3CA P42336 2/20 0.40
PIK3CB P42338 2/20 0.40
PIK3CG P48736 2/20 0.40
BTK Q06187 6/20 0.39
USP30 Q70CQ3 1/20 0.38
CHEK2 O96017 2/20 0.38
TNF P01375 2/20 0.38
LITAF Q99732 2/20 0.38
HDAC4 P56524 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
ATM Q13315 1/20 0.38
FGFR3 P22607 1/20 0.38
KDR P35968 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28456326 0.94 APLNR (0.42) APLNRPIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL28460224 0.92 CACNB4 (0.41) PIK3CDPIK3CAPIK3CBPIK3CGALDH1A1
SCHEMBL28450201 0.90 GPR119 (0.44) FGFR3KDRALDH1A1LMNA
SCHEMBL28452396 0.86 BTK (0.53) BTK
SCHEMBL28457726 0.86 PIK3CD (0.41) PIK3CDPIK3CAPIK3CBPIK3CGBTK
SCHEMBL28898962 0.85 CACNB4 (0.41) PIK3CDPIK3CAPIK3CBPIK3CGUSP30
SCHEMBL28452368 0.84 IRAK4 (0.43) ALDH1A1LMNA
SCHEMBL28455471 0.83 BTK (0.43) APLNRPIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL28898133 0.81 APLNR (0.44) APLNRPIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL28898960 0.81 GPR119 (0.46) PIK3CDPIK3CAPIK3CBPIK3CGUSP30

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111662232-B Small molecule compound with 2H-indazole structure and synthesis and application thereof 中国科学院上海药物研究所 2022-08-02 CN disclosed
CN-111662232-A Small molecule compound with 2H-indazole structure and synthesis and application thereof 中国科学院上海药物研究所 2020-09-15 CN disclosed