SCHEMBL28898155

SCHEMBL28898155

CC(C)(C)OC(=O)N1CCC(n2cc3cc(-c4ccccc4F)ccc3n2)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 3/20 0.45
JAK3 P52333 2/20 0.45
PTK2 Q05397 2/20 0.45
GPR119 Q8TDV5 8/20 0.45
JAK1 P23458 1/20 0.42
MET P08581 1/20 0.41
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
TSHR P16473 1/20 0.41
CRHBP P24387 1/20 0.41
HTT P42858 1/20 0.41
KMT2A Q03164 1/20 0.41
CRHR2 Q13324 1/20 0.41
HSD17B10 Q99714 1/20 0.41
BTK Q06187 1/20 0.41
TLR8 Q9NR97 1/20 0.41
MAPT P10636 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28455465 0.93 HSD17B13 (0.44) JAK2JAK3PTK2GPR119JAK1
SCHEMBL28457726 0.89 PIK3CD (0.41) JAK2JAK1BTK
SCHEMBL28450201 0.85 GPR119 (0.44) JAK2JAK3PTK2GPR119KDM4E
SCHEMBL25204156 0.82 GPR119 (0.44) JAK2JAK3PTK2GPR119MET
SCHEMBL28456262 0.82 PIK3CD (0.41) JAK2JAK1BTK
SCHEMBL28898961 0.82 BTK (0.47) BTKTLR8
SCHEMBL20135591 0.82 GPR119 (0.50) JAK2JAK3PTK2GPR119MET
SCHEMBL17096981 0.81 TDO2 (0.43) GPR119
SCHEMBL25204635 0.80 GPR119 (0.44) JAK2JAK3PTK2GPR119TLR8
SCHEMBL20134846 0.80 CNR1 (0.47) GPR119MEN1HPGDKMT2AHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111662232-B Small molecule compound with 2H-indazole structure and synthesis and application thereof 中国科学院上海药物研究所 2022-08-02 CN disclosed
CN-111662232-A Small molecule compound with 2H-indazole structure and synthesis and application thereof 中国科学院上海药物研究所 2020-09-15 CN disclosed