SCHEMBL28898960

SCHEMBL28898960

CC(C)(C)OC(=O)N1CCCC(n2cc3cc(-c4ccncc4)ccc3n2)C1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 5/20 0.46
USP30 Q70CQ3 3/20 0.43
CHEK2 O96017 2/20 0.42
CYP2C9 P11712 1/20 0.41
TLR8 Q9NR97 1/20 0.41
HCAR1 Q9BXC0 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
PTPN2 P17706 1/20 0.40
PTPN1 P18031 1/20 0.40
PTPN6 P29350 1/20 0.40
FPR2 P25090 1/20 0.40
PIK3CD O00329 2/20 0.39
PIK3CA P42336 2/20 0.39
PIK3CB P42338 2/20 0.39
PIK3CG P48736 2/20 0.39
FGFR3 P22607 1/20 0.39
KDR P35968 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28461486 0.93 GPR119 (0.46) GPR119USP30CHEK2CYP2C9HCAR1
SCHEMBL28450241 0.86 USP30 (0.50) GPR119USP30CHEK2HCAR1
SCHEMBL28463632 0.85 FPR2 (0.48) USP30CHEK2CYP2C9HCAR1HDAC4
SCHEMBL28457726 0.84 PIK3CD (0.41) USP30CHEK2HDAC4HDAC6PIK3CD
SCHEMBL28449733 0.83 CNR1 (0.46) GPR119USP30CHEK2HDAC4HDAC6
SCHEMBL28898963 0.83 HDAC1 (0.46) GPR119USP30CHEK2HDAC4HDAC6
SCHEMBL28458581 0.83 SRC (0.47) GPR119USP30CHEK2HDAC4HDAC6
SCHEMBL28458448 0.82 GPR119 (0.48) GPR119USP30CHEK2CYP2C9HDAC4
SCHEMBL29968466 0.82 GPR119 (0.48) GPR119USP30CHEK2CYP2C9HDAC4
SCHEMBL28456031 0.82 BTK (0.55)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111662232-B Small molecule compound with 2H-indazole structure and synthesis and application thereof 中国科学院上海药物研究所 2022-08-02 CN disclosed
CN-111662232-A Small molecule compound with 2H-indazole structure and synthesis and application thereof 中国科学院上海药物研究所 2020-09-15 CN disclosed