SCHEMBL28459351

SCHEMBL28459351

C=C(NC(=O)c1ccc(CCC)cc1)c1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 2/20 0.61
POLB P06746 3/20 0.59
CTDSP1 Q9GZU7 3/20 0.59
NPC1 O15118 2/20 0.59
RAB9A P51151 2/20 0.59
KMT2A Q03164 1/20 0.59
MCOLN3 Q8TDD5 1/20 0.59
GAA P10253 4/20 0.51
ALDH1A1 P00352 3/20 0.51
TRPV1 Q8NER1 2/20 0.51
KDM4E B2RXH2 1/20 0.51
HDAC1 Q13547 3/20 0.49
TMEM97 Q5BJF2 1/20 0.48
SIGMAR1 Q99720 1/20 0.48
THRB P10828 1/20 0.47
HDAC3 O15379 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
LMNA P02545 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28459349 0.91 TRPV1 (0.63) PLK1POLBCTDSP1NPC1RAB9A
SCHEMBL28465310 0.90 TRPV1 (0.58) PLK1KMT2AALDH1A1TRPV1HDAC1
SCHEMBL28469389 0.88 PLK1 (0.59) PLK1POLBCTDSP1NPC1RAB9A
SCHEMBL6551314 0.82 ALDH1A1 (0.55) CTDSP1NPC1RAB9AKMT2AGAA
SCHEMBL24534776 0.81 PLK1 (0.65) PLK1POLBCTDSP1NPC1RAB9A
SCHEMBL28466726 0.81 PLK1 (0.54) PLK1POLBCTDSP1NPC1RAB9A
SCHEMBL28463608 0.79 CCR6 (0.59) POLBNPC1RAB9AKMT2AGAA
SCHEMBL28459281 0.78 MEN1 (0.67) PLK1POLBNPC1RAB9AKMT2A
SCHEMBL28459686 0.78 PLK1 (0.62) PLK1POLBNPC1RAB9AKMT2A
SCHEMBL13670699 0.77 PLK1 (0.73) PLK1POLBCTDSP1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111747904-A Polyfluoroalkenyl substituted oxazole compound and preparation method thereof 南京工业大学 2020-10-09 CN claimed
CN-111747904-A Polyfluoroalkenyl substituted oxazole compound and preparation method thereof 南京工业大学 2020-10-09 CN disclosed