SCHEMBL28465310

SCHEMBL28465310

C=C(NC(=O)c1ccc(CCCCC)cc1)c1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.58
PLK1 P53350 5/20 0.57
PLK3 Q9H4B4 4/20 0.56
THRA P10827 3/20 0.54
THRB P10828 3/20 0.54
RARB P10826 5/20 0.52
HDAC1 Q13547 1/20 0.52
MEN1 O00255 1/20 0.51
ALDH1A1 P00352 1/20 0.51
RARA P10276 1/20 0.51
MAPT P10636 1/20 0.51
MTOR P42345 1/20 0.51
KMT2A Q03164 1/20 0.51
HAO1 Q9UJM8 1/20 0.51
HDAC8 Q9BY41 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28459349 0.96 TRPV1 (0.63) TRPV1PLK1PLK3THRATHRB
SCHEMBL28459351 0.90 PLK1 (0.61) TRPV1PLK1THRBHDAC1ALDH1A1
SCHEMBL28469389 0.84 PLK1 (0.59) TRPV1PLK1HDAC1ALDH1A1KMT2A
SCHEMBL24534632 0.83 PLK1 (0.60) TRPV1PLK1PLK3THRATHRB
SCHEMBL28460406 0.82 THRA (0.63) PLK1THRATHRBRARBMEN1
SCHEMBL24534900 0.82 HAO1 (0.59) TRPV1PLK1PLK3THRATHRB
SCHEMBL28463607 0.81 NR1H4 (0.59) PLK1RARBMEN1KMT2A
SCHEMBL28462599 0.81 MEN1 (0.60) PLK1MEN1ALDH1A1MAPTKMT2A
SCHEMBL10602808 0.79 THRA (0.57) TRPV1THRATHRBRARBMEN1
SCHEMBL11227652 0.79 RARB (0.65) TRPV1THRATHRBRARBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111747904-A Polyfluoroalkenyl substituted oxazole compound and preparation method thereof 南京工业大学 2020-10-09 CN claimed
CN-111747904-A Polyfluoroalkenyl substituted oxazole compound and preparation method thereof 南京工业大学 2020-10-09 CN disclosed