SCHEMBL7705613

SCHEMBL7705613

c1ccc2c(c1)CCN=C2c1cnccn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 2/20 0.45
NOS2 P35228 1/20 0.45
ADRA1A P35348 2/20 0.43
ADRA1B P35368 2/20 0.43
ADRA1D P25100 1/20 0.42
CYP19A1 P11511 6/20 0.42
CYP11B2 P19099 6/20 0.42
MAOA P21397 1/20 0.41
NISCH Q9Y2I1 1/20 0.39
CYP11B1 P15538 5/20 0.37
CYP2D6 P10635 4/20 0.37
HRH1 P35367 4/20 0.37
CHRM1 P11229 1/20 0.37
HTR2A P28223 1/20 0.37
KCNH2 Q12809 1/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP17A1 P05093 1/20 0.36
CYP3A4 P08684 1/20 0.35
METAP2 P50579 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7701012 0.82 NOS3 (0.49) NOS3NOS2ADRA1AADRA1BADRA1D
SCHEMBL7697911 0.78 NOS3 (0.45) NOS3NOS2CYP19A1CYP11B2MAOA
SCHEMBL30920956 0.77 CYP2A6 (0.40) NOS3NOS2ADRA1AMAOANISCH
SCHEMBL7705661 0.77 NOS3 (0.44) NOS3NOS2MAOAKDM4EALDH1A1
SCHEMBL31083746 0.76 CYP11B1 (0.54) NOS3NOS2CYP19A1CYP11B2NISCH
SCHEMBL29537716 0.76 CYP11B1 (0.54) NOS3NOS2CYP19A1CYP11B2NISCH
SCHEMBL10426776 0.76 ADRB2 (0.48) ADRA1AADRA1BADRA1DCYP11B2MAOA
SCHEMBL7699089 0.76 NOS3 (0.49) NOS3NOS2CYP19A1CYP11B2MAOA
SCHEMBL7704052 0.75 GRIN2D (0.45) NOS3NOS2ADRA1AADRA1BADRA1D
SCHEMBL7698058 0.74 NOS3 (0.44) NOS3NOS2MAOACYP2D6KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0901488-B1 2,4-DIAMINOPYRIMIDINE DERIVATIVES BASILEA PHARMACEUTICA AG (CH) 2002-11-06 EP disclosed
EP-0901488-A1 2,4-DIAMINOPYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1999-03-17 EP disclosed
US-5866583-A Substituted 2,4-diaminopyrimidines HOFFMANN-LA ROCHE INC. (US) 1999-02-02 US disclosed
WO-1997043277-A1 2,4-DIAMINOPYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1997-11-20 WO disclosed