SCHEMBL2846211

SCHEMBL2846211

CC[Si](CC)(CC)OC(C)(C)C(F)(F)CC(=O)O

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 1/20 0.35
CHRM1 P11229 1/20 0.35
TBXA2R P21731 1/20 0.35
ADRA1A P35348 1/20 0.35
CYP2D6 P10635 1/20 0.34
TSHR P16473 1/20 0.34
CYP2C19 P33261 1/20 0.34
HIF1A Q16665 1/20 0.34
FFAR3 O14843 1/20 0.32
KDM4E B2RXH2 1/20 0.31
FFAR1 O14842 1/20 0.31
CPT2 P23786 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
ALDH1A1 P00352 1/20 0.31
ACLY P53396 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31507719 0.73 KCNN4 (0.35) CYP2C19HIF1AALDH1A1
SCHEMBL2846165 0.71 HMGCR (0.34) HMGCRCHRM1TBXA2RADRA1ACYP2D6
SCHEMBL10385551 0.68 HMGCR (0.50) HMGCRCHRM1TBXA2RADRA1ACYP2D6
SCHEMBL3179512 0.68 NAALAD2 (0.37) FFAR3ALDH1A1
SCHEMBL9438232 0.67 ACLY (0.48) HMGCRCHRM1TBXA2RADRA1ACYP2D6
SCHEMBL2851193 0.65 ALDH1A1 (0.38) TSHRHIF1AFFAR3FFAR1TDP1
SCHEMBL28665121 0.65 ACLY (0.46) HMGCRCHRM1TBXA2RADRA1ACYP2D6
SCHEMBL11227427 0.62 ACLY (0.44) HMGCRCHRM1TBXA2RADRA1ACYP2D6
SCHEMBL865358 0.62 ACLY (0.44) HMGCRCHRM1TBXA2RADRA1ACYP2D6
SCHEMBL16269785 0.62

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2025667-B1 9,10-SECOPREGNANE DERIVATIVE AND PHARMACEUTICAL NIPPON SHINYAKU CO LTD (JP) 2016-08-10 EP disclosed
US-8796246-B2 9, 10-secopregnane derivative and pharmaceutical NIPPON SHINYAKU CO., LTD. (JP) 2014-08-05 US disclosed
US-20100130454-A1 9,10-SECOPREGNANE DERIVATIVES AND MEDICINE NIPPON SHINYAKU CO., LTD. (JP) 2010-05-27 US disclosed
US-20100016263-A1 9, 10-SECOPREGNANE DERIVATIVE AND PHARMACEUTICAL NIPPON SHINYAKU CO., LTD. (JP) 2010-01-21 US disclosed
EP-2025667-A1 9,10-SECOPREGNANE DERIVATIVE AND PHARMACEUTICAL Nippon Shinyaku Co., Ltd. (JP) 2009-02-18 EP disclosed
EP-1829860-A1 9,10-SECOPREGNANE DERIVATIVE AND MEDICINE Nippon Shinyaku Co., Ltd. (JP) 2007-09-05 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100130454-A1 9,10-SECOPREGNANE DERIVATIVES AND MEDICINE VDR, CYP2R1, CYP24A1 HMGCR 367/4885CHRM1 403/4885TBXA2R 372/4885
US-20100016263-A1 9, 10-SECOPREGNANE DERIVATIVE AND PHARMACEUTICAL CYP2R1, VDR, CYP24A1 HMGCR 309/4885CHRM1 500/4885TBXA2R 422/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.