SCHEMBL28463285

SCHEMBL28463285

O=C(O)C(=Cc1ccccc1)/C=C/c1ccc(Br)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1B1 Q16678 2/20 0.58
HDAC3 O15379 2/20 0.49
HDAC4 P56524 2/20 0.49
HDAC1 Q13547 2/20 0.49
HDAC2 Q92769 2/20 0.49
HDAC8 Q9BY41 2/20 0.49
HDAC6 Q9UBN7 2/20 0.49
MAPT P10636 4/20 0.48
LMNA P02545 3/20 0.48
ALDH1A1 P00352 3/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
CYP1A2 P05177 2/20 0.48
CYP2D6 P10635 2/20 0.48
TNKS O95271 1/20 0.48
HCAR2 Q8TDS4 1/20 0.48
HDAC7 Q8WUI4 1/20 0.48
HDAC10 Q969S8 1/20 0.48
HDAC11 Q96DB2 1/20 0.48
TNKS2 Q9H2K2 1/20 0.48
HDAC9 Q9UKV0 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28461467 1.00 CYP1B1 (0.58) CYP1B1HDAC3HDAC4HDAC1HDAC2
SCHEMBL2981331 0.89 MAPT (0.59) CYP1B1HDAC3HDAC4HDAC1HDAC2
SCHEMBL28468276 0.83 CYP1B1 (0.51) CYP1B1HDAC3HDAC4HDAC1HDAC2
SCHEMBL28468278 0.83 CYP1B1 (0.51) CYP1B1HDAC3HDAC4HDAC1HDAC2
SCHEMBL12144576 0.80 LMNA (0.76) CYP1B1HDAC3HDAC4HDAC1HDAC2
SCHEMBL7167809 0.78 MAPT (0.59) CYP1B1HDAC3HDAC4HDAC1HDAC2
SCHEMBL29466710 0.78 MAPT (0.56) CYP1B1HDAC3HDAC4HDAC1HDAC2
SCHEMBL3469448 0.78 MMP1 (0.60) HDAC3HDAC4HDAC1HDAC2HDAC8
SCHEMBL6212312 0.77 CYP1B1 (0.54) CYP1B1HDAC3HDAC4HDAC1HDAC2
SCHEMBL15486079 0.77 MAPT (0.57) CYP1B1HDAC3HDAC4HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109970560-B Preparation method of tri-substituted 1, 3-diene compound 南京工业大学 2020-09-29 CN disclosed