SCHEMBL28468477

SCHEMBL28468477

O=C(NO)c1ccc(CN2C(=O)C(=O)c3cc(Cl)ccc32)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH3A1 P30838 5/20 0.64
ALDH1A1 P00352 1/20 0.64
ALDH2 P05091 1/20 0.64
HDAC1 Q13547 9/20 0.62
HDAC6 Q9UBN7 8/20 0.62
HDAC8 Q9BY41 7/20 0.62
HDAC7 Q8WUI4 4/20 0.56
ACHE P22303 1/20 0.54
CA12 O43570 1/20 0.54
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
CA9 Q16790 1/20 0.54
HDAC2 Q92769 4/20 0.54
HDAC3 O15379 3/20 0.54
HDAC4 P56524 3/20 0.54
HDAC10 Q969S8 3/20 0.54
HDAC11 Q96DB2 3/20 0.54
HDAC9 Q9UKV0 3/20 0.54
HDAC5 Q9UQL6 3/20 0.54
CES2 O00748 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28799598 0.88 ALDH3A1 (0.65) ALDH3A1ALDH1A1ALDH2HDAC1HDAC6
SCHEMBL28464687 0.88 ACHE (0.73) ALDH3A1ALDH1A1ALDH2HDAC1HDAC6
SCHEMBL28469301 0.86 HDAC1 (0.55) ALDH3A1ALDH1A1ALDH2HDAC1HDAC6
SCHEMBL28470163 0.84 ALDH3A1 (0.62) ALDH3A1ALDH1A1ALDH2ACHECA12
SCHEMBL29869527 0.84 ALDH3A1 (0.82) ALDH3A1ALDH1A1ALDH2ACHECA12
SCHEMBL11186018 0.84 ALDH3A1 (0.82) ALDH3A1ALDH1A1ALDH2ACHECA12
SCHEMBL28462499 0.83 HDAC1 (0.72) ALDH3A1ALDH1A1ALDH2HDAC1HDAC6
SCHEMBL29699570 0.82 CASP3 (0.67) ALDH1A1HDAC1HDAC6HDAC8HDAC7
SCHEMBL28799594 0.82 CASP3 (0.67) ALDH1A1HDAC1HDAC6HDAC8HDAC7
SCHEMBL30387645 0.80 APAF1 (0.57) ALDH3A1ALDH1A1ALDH2ACHECA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111747883-B 1-benzyl isatin derivative and synthesis method and application thereof 中南大学 2022-07-01 CN disclosed
CN-111747883-A 1-benzyl isatin derivative and synthesis method and application thereof 中南大学 2020-10-09 CN disclosed