SCHEMBL2847273

SCHEMBL2847273

Cc1cccc(-c2c(Cl)cccc2C(=O)C2CCCN(C(=O)O)C2)c1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.47
RHOA P61586 1/20 0.44
GRM5 P41594 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
ALDH1A1 P00352 2/20 0.42
HSD11B1 P28845 5/20 0.42
KDM2B Q8NHM5 2/20 0.42
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2846275 0.87 POLB (0.45) POLBRHOAMEN1KMT2AALDH1A1
SCHEMBL2849948 0.87 POLB (0.45) POLBRHOAMEN1KMT2AALDH1A1
SCHEMBL2850274 0.86 KAT6A (0.49) POLBRHOAMEN1KMT2AALDH1A1
SCHEMBL2850273 0.86 KAT6A (0.49) POLBRHOAMEN1KMT2AALDH1A1
SCHEMBL5592323 0.84 POLB (0.42) POLBRHOAGRM5MEN1KMT2A
SCHEMBL5604174 0.83 POLB (0.43) POLBMEN1KMT2AALDH1A1KDM2B
SCHEMBL3963250 0.78 HPGD (0.56) POLBRHOAMEN1KMT2AALDH1A1
SCHEMBL4755206 0.77 POLB (0.52) POLBMEN1KMT2AALDH1A1KDM2B
SCHEMBL4748847 0.77 KAT7 (0.44)
SCHEMBL2850721 0.77 MEN1 (0.41) POLBMEN1KMT2AALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100130471-A1 Renin Inhibitors SMITHKLINE BEECHAM CORPORATION 2010-05-27 US disclosed
EP-2167609-A1 RENIN INHIBITORS Vitae Pharmaceuticals, Inc. (US) 2010-03-31 EP disclosed
WO-2009096996-A1 RENIN INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2009-08-06 WO disclosed
WO-2008124575-A1 RENIN INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-10-16 WO disclosed
WO-2008124577-A1 RENIN INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-10-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100130471-A1 Renin Inhibitors ACE, REN, DNPEP POLB 1262/4885RHOA 2661/4885GRM5 1565/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.