SCHEMBL28477374

SCHEMBL28477374

COCCC(C(=O)OC)(C(=O)OC(C)(C)C)c1ccnc(NS(=O)(=O)CCc2ccc(OC)cc2)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP6 P55212 1/20 0.41
GAA P10253 2/20 0.39
MMP8 P22894 1/20 0.38
MMP12 P39900 1/20 0.38
MMP13 P45452 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CTPS1 P17812 3/20 0.35
AR P10275 1/20 0.35
PTPN1 P18031 1/20 0.34
PTPN11 Q06124 1/20 0.34
PTPN22 Q9Y2R2 1/20 0.34
EDNRB P24530 1/20 0.33
EDNRA P25101 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
NR3C2 P08235 1/20 0.33
PTPRB P23467 1/20 0.33
POLB P06746 1/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21384619 0.87 CASP6 (0.44) CASP6GAAMMP8MMP12MMP13
SCHEMBL21392311 0.83 CTPS1 (0.47) MEN1KMT2ACTPS1ARHPGD
SCHEMBL21373726 0.79 CTPS1 (0.45) CTPS1
SCHEMBL21392152 0.79 PTPN1 (0.36) MMP13PTPN1
SCHEMBL30415860 0.79 PTPN1 (0.36) MMP13PTPN1
SCHEMBL26977404 0.79 AR (0.35) CASP6GAAMEN1KMT2AAR
SCHEMBL21392150 0.76 RAB9A (0.32) GAAKMT2AARRAB9APOLB
SCHEMBL21373801 0.73 AAK1 (0.36) CTPS1
SCHEMBL28478417 0.73 CASP6 (0.42) CASP6GAAMMP8MMP12MMP13
SCHEMBL21387592 0.71 CTPS1 (0.31) CTPS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111868051-B Aminopyrimidine derivatives as CTPS1 inhibitors 斯泰普制药股份公司 2024-04-09 CN disclosed
CN-111868051-A Aminopyrimidine derivatives as CTPS1 inhibitors 斯泰普制药股份公司 2020-10-30 CN disclosed