SCHEMBL28479671

SCHEMBL28479671

CC1(C)OB(c2ccc3oc(NS(C)(=O)=O)nc3c2)OC1(C)C

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
CA9 Q16790 2/20 0.43
CA12 O43570 1/20 0.43
CA3 P07451 1/20 0.43
CA4 P22748 1/20 0.43
CA6 P23280 1/20 0.43
CA5A P35218 1/20 0.43
CA7 P43166 1/20 0.43
CA14 Q9ULX7 1/20 0.43
CA5B Q9Y2D0 1/20 0.43
FBP1 P09467 17/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7899481 0.80 PIK3CA (0.45) CA1CA2CA9
SCHEMBL13370383 0.78 POLB (0.35) CA1CA2CA9CA12CA3
SCHEMBL3478062 0.78 NPC1 (0.54)
SCHEMBL18613753 0.77 HDAC6 (0.38)
SCHEMBL3534341 0.76 L3MBTL1 (0.46)
SCHEMBL3478060 0.75 HDAC6 (0.53)
SCHEMBL2724794 0.74 LMNA (0.49) CA1CA2CA9CA12CA3
SCHEMBL29867543 0.74 LMNA (0.49) CA1CA2CA9CA12CA3
SCHEMBL17378988 0.73 CA1 (0.47) CA1CA2CA9CA12CA3
SCHEMBL22160380 0.72 LPL (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111848629-B mTOR/HDAC dual inhibitor and application thereof 安徽中医药大学 2021-06-11 CN disclosed
CN-111848629-A mTOR/HDAC dual inhibitor and application thereof 安徽中医药大学 2020-10-30 CN disclosed