SCHEMBL2848312

SCHEMBL2848312

O=C(NCCc1ccccc1)c1cnn(-c2ccc([N+](=O)[O-])cc2)c1C(F)(F)F

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.56
MAPT P10636 6/20 0.56
ALDH1A1 P00352 2/20 0.55
KDM4E B2RXH2 1/20 0.55
SMN1; SMN2 Q16637 3/20 0.55
NPC1 O15118 2/20 0.55
RAB9A P51151 2/20 0.55
TAAR1 Q96RJ0 1/20 0.55
POLB P06746 1/20 0.49
ACHE P22303 3/20 0.49
DDR1 Q08345 1/20 0.49
MAPK11 Q15759 1/20 0.49
MAPK14 Q16539 1/20 0.49
DDR2 Q16832 1/20 0.49
TMEM97 Q5BJF2 1/20 0.49
MAP3K20 Q9NYL2 1/20 0.49
MAP3K2 Q9Y2U5 1/20 0.49
GSK3B P49841 1/20 0.48
NPSR1 Q6W5P4 1/20 0.47
KMT2A Q03164 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2855062 0.90 CCR1 (0.65) CCR1MAPTALDH1A1KDM4ESMN1; SMN2
SCHEMBL2852043 0.89 KDM4E (0.70) CCR1MAPTALDH1A1KDM4ESMN1; SMN2
SCHEMBL2859017 0.87 MAPT (0.69) CCR1MAPTALDH1A1KDM4ESMN1; SMN2
SCHEMBL2858927 0.87 KDM4E (0.61) CCR1MAPTALDH1A1KDM4ESMN1; SMN2
SCHEMBL2853014 0.86 KDM4E (0.60) CCR1MAPTALDH1A1KDM4ESMN1; SMN2
SCHEMBL2854304 0.84 NPC1 (0.49) CCR1MAPTALDH1A1KDM4ESMN1; SMN2
SCHEMBL2850321 0.84 SMN1; SMN2 (0.47) CCR1MAPTALDH1A1KDM4ESMN1; SMN2
SCHEMBL24304030 0.83 TRPC3 (0.60) CCR1MAPTALDH1A1KDM4ESMN1; SMN2
SCHEMBL2855239 0.83 ALDH1A1 (0.56) MAPTALDH1A1KDM4ESMN1; SMN2NPC1
SCHEMBL2857175 0.82 MAPT (0.57) CCR1MAPTALDH1A1KDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed