SCHEMBL2853014

SCHEMBL2853014

O=C(NCCc1ccccc1)c1cnn(-c2ccc(Cl)cc2)c1C(F)(F)F

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.60
ALDH1A1 P00352 1/20 0.60
MAPT P10636 5/20 0.57
ABCB1 P08183 1/20 0.53
CCR1 P32246 3/20 0.53
POLB P06746 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
HSP90AA1 P07900 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
P2RX7 Q99572 1/20 0.52
DDR1 Q08345 1/20 0.51
MAPK11 Q15759 1/20 0.51
MAPK14 Q16539 1/20 0.51
DDR2 Q16832 1/20 0.51
TMEM97 Q5BJF2 1/20 0.51
MAP3K20 Q9NYL2 1/20 0.51
MAP3K2 Q9Y2U5 1/20 0.51
LMNA P02545 2/20 0.51
TRPC3 Q13507 1/20 0.51
CCNA2 P20248 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2852043 0.92 KDM4E (0.70) KDM4EALDH1A1MAPTCCR1POLB
SCHEMBL2859017 0.90 MAPT (0.69) KDM4EALDH1A1MAPTCCR1POLB
SCHEMBL2858927 0.90 KDM4E (0.61) KDM4EALDH1A1MAPTCCR1POLB
SCHEMBL2852015 0.89 CCR1 (0.63) KDM4EALDH1A1MAPTCCR1POLB
SCHEMBL13513697 0.89 ABCB1 (0.58) KDM4EALDH1A1MAPTABCB1CCR1
SCHEMBL2857175 0.88 MAPT (0.57) KDM4EALDH1A1MAPTCCR1POLB
SCHEMBL2855239 0.87 ALDH1A1 (0.56) KDM4EALDH1A1MAPTPOLBSMN1; SMN2
SCHEMBL2856467 0.86 P2RX7 (0.51) KDM4EALDH1A1MAPTCCR1SMN1; SMN2
SCHEMBL2848312 0.86 CCR1 (0.56) KDM4EALDH1A1MAPTCCR1POLB
SCHEMBL2855315 0.85 KDM4E (0.65) KDM4EALDH1A1MAPTCCR1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed