SCHEMBL2855239

SCHEMBL2855239

COc1ccc(-n2ncc(C(=O)NCCc3ccccc3)c2C(F)(F)F)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.56
KDM4E B2RXH2 4/20 0.56
MAPT P10636 7/20 0.54
DGAT2 Q96PD7 1/20 0.51
KMT2A Q03164 3/20 0.51
SMN1; SMN2 Q16637 3/20 0.50
POLB P06746 1/20 0.50
DDR1 Q08345 1/20 0.49
MAPK11 Q15759 1/20 0.49
MAPK14 Q16539 1/20 0.49
DDR2 Q16832 1/20 0.49
TMEM97 Q5BJF2 1/20 0.49
MAP3K20 Q9NYL2 1/20 0.49
MAP3K2 Q9Y2U5 1/20 0.49
TP53 P04637 2/20 0.49
HPGD P15428 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
GAA P10253 2/20 0.48
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2850316 0.90 TP53 (0.59) ALDH1A1KDM4EMAPTDGAT2SMN1; SMN2
SCHEMBL2852043 0.90 KDM4E (0.70) ALDH1A1KDM4EMAPTKMT2ASMN1; SMN2
SCHEMBL2858927 0.88 KDM4E (0.61) ALDH1A1KDM4EMAPTSMN1; SMN2POLB
SCHEMBL2859017 0.88 MAPT (0.69) ALDH1A1KDM4EMAPTSMN1; SMN2POLB
SCHEMBL2853014 0.87 KDM4E (0.60) ALDH1A1KDM4EMAPTSMN1; SMN2POLB
SCHEMBL2851942 0.85 NPC1 (0.64) ALDH1A1KDM4EMAPTKMT2ASMN1; SMN2
SCHEMBL2852633 0.84 TAAR1 (0.57) ALDH1A1KDM4EMAPTKMT2ATP53
SCHEMBL10366447 0.84 TRPC3 (0.62) ALDH1A1KDM4EMAPTDGAT2KMT2A
SCHEMBL26965090 0.84 ALDH1A1 (0.50) ALDH1A1KDM4EMAPTDGAT2KMT2A
SCHEMBL2848312 0.83 CCR1 (0.56) ALDH1A1KDM4EMAPTKMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed