SCHEMBL28498296

SCHEMBL28498296

CCc1ccc2c(c1)C(=O)C(C(F)(F)C(F)(F)C(F)(F)C(F)(F)F)CC2

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.33
DRD2 P14416 2/20 0.33
HTR2A P28223 2/20 0.33
HTR2C P28335 2/20 0.33
HTR2B P41595 2/20 0.33
NPC1 O15118 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
MAPK1 P28482 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
DRD1 P21728 1/20 0.33
CYP19A1 P11511 2/20 0.33
GPR119 Q8TDV5 1/20 0.32
PDK2 Q15119 1/20 0.31
CYP27A1 Q02318 1/20 0.31
CYP24A1 Q07973 1/20 0.31
KDM4E B2RXH2 1/20 0.30
CYP1A2 P05177 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28505292 0.87 S1PR1 (0.37) DRD2HTR2AHTR2CCYP2C19
SCHEMBL28505200 0.84 PARP11 (0.38) DRD2HTR2AHTR2CHTR2BCYP19A1
SCHEMBL28507951 0.83 ACHE (0.43) ALDH1A1NPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL28500672 0.82 TYMS (0.39) MAPTL3MBTL1CYP19A1PDK2
SCHEMBL28507112 0.82 ACHE (0.43) DRD2HTR2AHTR2CHTR2BSIGMAR1
SCHEMBL28504434 0.81 PARP1 (0.35) ALDH1A1DRD2HTR2AHTR2CHTR2B
SCHEMBL28496512 0.81 DRD2 (0.35) DRD2HTR2APDK2
SCHEMBL28508889 0.81 F7 (0.39) HTR2AHTR2CMAPTMAPK1
SCHEMBL28507925 0.81 PBRM1 (0.46) DRD2CYP19A1
SCHEMBL28905422 0.81 PARP10 (0.39) MAPK1L3MBTL1CYP19A1CYP1A2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112159411-A Trifluoromethyl substituted pyrimido [1,3] diaza compound and preparation method thereof 南京工业大学 2021-01-01 CN claimed
CN-112159411-A Trifluoromethyl substituted pyrimido [1,3] diaza compound and preparation method thereof 南京工业大学 2021-01-01 CN disclosed