SCHEMBL28905422

SCHEMBL28905422

O=C1c2cc(Br)ccc2CCC1C(F)(F)C(F)(F)C(F)(F)C(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PARP10 Q53GL7 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PARP1 P09874 1/20 0.39
TYMS P04818 2/20 0.32
ADRA2A P08913 1/20 0.32
PNMT P11086 1/20 0.32
CYP19A1 P11511 1/20 0.32
METAP1 P53582 1/20 0.31
S100A4 P26447 1/20 0.31
CYP1A2 P05177 1/20 0.31
MAPK1 P28482 1/20 0.31
TDP2 O95551 1/20 0.31
PARP11 Q9NR21 1/20 0.31
PBRM1 Q86U86 1/20 0.30
SRD5A1 P18405 1/20 0.30
DDB1 Q16531 1/20 0.30
CRBN Q96SW2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28507925 0.86 PBRM1 (0.46) TYMSCYP19A1PBRM1CRBN
SCHEMBL28507112 0.85 ACHE (0.43) PARP10PARP1TYMSSRD5A1DDB1
SCHEMBL28507951 0.84 ACHE (0.43) PARP10PARP1TYMSMETAP1PARP11
SCHEMBL28501370 0.84 TDP2 (0.33) TYMSPNMTTDP2SRD5A1
SCHEMBL28508889 0.84 F7 (0.39) PARP10PARP1TYMSPNMTMETAP1
SCHEMBL28496512 0.84 DRD2 (0.35) TYMSDDB1CRBN
SCHEMBL28504434 0.82 PARP1 (0.35) PARP10L3MBTL1PARP1CYP19A1SRD5A1
SCHEMBL28498301 0.81 TYRO3 (0.39) PARP10L3MBTL1TDP2PARP11
SCHEMBL28501373 0.81 CYP19A1 (0.47) CYP19A1METAP1
SCHEMBL28500637 0.80 CYP19A1 (0.42) TDP1CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110003187-B Polyfluoroalkyl substituted benzofuran compound and preparation method thereof 南京工业大学 2021-11-05 CN claimed
CN-112159411-A Trifluoromethyl substituted pyrimido [1,3] diaza compound and preparation method thereof 南京工业大学 2021-01-01 CN claimed
CN-110003187-B Polyfluoroalkyl substituted benzofuran compound and preparation method thereof 南京工业大学 2021-11-05 CN disclosed
CN-112159411-A Trifluoromethyl substituted pyrimido [1,3] diaza compound and preparation method thereof 南京工业大学 2021-01-01 CN disclosed