SCHEMBL28507112

SCHEMBL28507112

O=C1c2cc(F)ccc2CCC1C(F)(F)C(F)(F)C(F)(F)C(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.43
PARP1 P09874 1/20 0.40
PARP10 Q53GL7 1/20 0.40
SRD5A1 P18405 5/20 0.36
TYMS P04818 2/20 0.33
AKR1A1 P14550 3/20 0.32
AKR1B1 P15121 3/20 0.32
DRD2 P14416 2/20 0.31
HTR2A P28223 2/20 0.31
HTR2C P28335 1/20 0.31
HTR2B P41595 1/20 0.31
SIGMAR1 Q99720 1/20 0.31
DDB1 Q16531 1/20 0.31
CRBN Q96SW2 1/20 0.31
KDM1A O60341 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28508889 0.85 F7 (0.39) PARP1PARP10SRD5A1TYMSHTR2A
SCHEMBL28507925 0.85 PBRM1 (0.46) TYMSAKR1B1DRD2CRBN
SCHEMBL28507951 0.85 ACHE (0.43) ACHEPARP1PARP10SRD5A1TYMS
SCHEMBL28496512 0.85 DRD2 (0.35) TYMSDRD2HTR2ADDB1CRBN
SCHEMBL28905422 0.85 PARP10 (0.39) PARP1PARP10SRD5A1TYMSDDB1
SCHEMBL28501370 0.85 TDP2 (0.33) SRD5A1TYMS
SCHEMBL28504434 0.83 PARP1 (0.35) PARP1PARP10SRD5A1DRD2HTR2A
SCHEMBL28498296 0.82 ALDH1A1 (0.33) DRD2HTR2AHTR2CHTR2BSIGMAR1
SCHEMBL28498134 0.82 HPGD (0.36)
SCHEMBL28500637 0.81 CYP19A1 (0.42) ACHEDRD2HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110003187-B Polyfluoroalkyl substituted benzofuran compound and preparation method thereof 南京工业大学 2021-11-05 CN claimed
CN-112159411-A Trifluoromethyl substituted pyrimido [1,3] diaza compound and preparation method thereof 南京工业大学 2021-01-01 CN claimed
CN-110003187-B Polyfluoroalkyl substituted benzofuran compound and preparation method thereof 南京工业大学 2021-11-05 CN disclosed
CN-112159411-A Trifluoromethyl substituted pyrimido [1,3] diaza compound and preparation method thereof 南京工业大学 2021-01-01 CN disclosed