SCHEMBL28499404

SCHEMBL28499404

NC(=O)c1cc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(-c4ccc(C(F)(F)F)cc4)c3)c(F)c2)ccn1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 5/20 0.62
BRAF P15056 11/20 0.62
KDR P35968 10/20 0.62
MAPK14 Q16539 5/20 0.62
RIPK2 O43353 2/20 0.62
ABCB11 O95342 2/20 0.62
ABL1 P00519 2/20 0.62
RET P07949 2/20 0.62
HTR1A P08908 2/20 0.62
PDGFRB P09619 2/20 0.62
ADORA3 P0DMS8 2/20 0.62
KIT P10721 2/20 0.62
FGFR1 P11362 2/20 0.62
PDGFRA P16234 2/20 0.62
FLT1 P17948 2/20 0.62
MAOA P21397 2/20 0.62
EPHA1 P21709 2/20 0.62
TBXA2R P21731 2/20 0.62
EPHA2 P29317 2/20 0.62
TTK P33981 2/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29643339 0.86 RAF1 (0.82) RAF1BRAFKDRMAPK14RIPK2
SCHEMBL432444 0.86 RAF1 (0.82) RAF1BRAFKDRMAPK14RIPK2
SCHEMBL28499406 0.86 RAF1 (0.66) RAF1BRAFKDRMAPK14RIPK2
SCHEMBL1662209 0.86 BRAF (0.69) RAF1BRAFKDRMAPK14RIPK2
SCHEMBL1661022 0.82 RAF1 (0.74) RAF1BRAFKDRMAPK14RIPK2
SCHEMBL1662217 0.81 BRAF (0.68) BRAFKDRMAPK14
SCHEMBL1662296 0.79 RAF1 (0.64) RAF1BRAFKDRMAPK14ABL1
SCHEMBL12333608 0.79 RAF1 (0.82) RAF1BRAFKDRMAPK14RIPK2
SCHEMBL1660260 0.79 MAPK14 (0.60) RAF1BRAFKDRMAPK14RIPK2
SCHEMBL4609009 0.78 BRAF (0.82) RAF1BRAFKDRMAPK14RIPK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112159351-B Preparation method of multi-target antitumor drug 广州南鑫药业有限公司 2021-12-07 CN disclosed
CN-112587485-A Medicine solid dispersion and preparation method thereof 湖南南新制药股份有限公司 2021-04-02 CN disclosed
CN-112159351-A Preparation method of multi-target antitumor drug 广州南鑫药业有限公司 2021-01-01 CN disclosed