SCHEMBL28499600

SCHEMBL28499600

Cc1cc(B2OC(C)(C)C(C)(C)O2)cc(C)c1N1CCN(CCO)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
LMNA P02545 1/20 0.36
DRD2 P14416 1/20 0.35
DRD3 P35462 1/20 0.35
NSD2 O96028 1/20 0.34
PABPC1 P11940 1/20 0.34
TP53 P04637 1/20 0.34
MAPT P10636 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
KDM4E B2RXH2 1/20 0.33
KCNJ5 P48544 1/20 0.33
KCNJ3 P48549 1/20 0.33
HTR7 P34969 2/20 0.33
OPRM1 P35372 1/20 0.33
OPRK1 P41145 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28906218 0.89 KCNJ5 (0.36) ALDH1A1MEN1KMT2ALMNADRD2
SCHEMBL28509585 0.89 ALDH1A1 (0.33) ALDH1A1MEN1KMT2AMAPTSMN1; SMN2
SCHEMBL24723411 0.83 LPL (0.33) ALDH1A1MEN1KMT2AMAPTSMN1; SMN2
SCHEMBL586151 0.78 LPL (0.41) ALDH1A1MEN1KMT2ADRD2DRD3
SCHEMBL24269630 0.77 ALDH1A1 (0.39) ALDH1A1MEN1KMT2ATP53MAPT
SCHEMBL18621693 0.77 DRD2 (0.45) DRD2DRD3OPRM1
SCHEMBL3665155 0.76 MEN1 (0.42) ALDH1A1MEN1KMT2ADRD2CYP3A4
SCHEMBL24722841 0.76 HRH4 (0.35) DRD2DRD3MAPTKDM4E
SCHEMBL13958134 0.75 DRD2 (0.38) ALDH1A1MEN1KMT2ADRD2DRD3
SCHEMBL24722942 0.75 ROCK1 (0.37) ALDH1A1MEN1KMT2AMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112243439-A Pyrrolo [2,3-B ] pyridines or pyrrolo [2,3-B ] pyrazines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-01-19 CN disclosed