SCHEMBL28906218

SCHEMBL28906218

Cc1cc(B2OC(C)(C)C(C)(C)O2)cc(C#N)c1N1CCN(CCO)CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNJ5 P48544 1/20 0.36
KCNJ3 P48549 1/20 0.36
LMNA P02545 3/20 0.34
ALDH1A1 P00352 3/20 0.34
KHK P50053 1/20 0.34
HTR7 P34969 2/20 0.33
GAA P10253 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
KDM4E B2RXH2 2/20 0.32
PKM P14618 2/20 0.32
TSHR P16473 1/20 0.32
MAPK1 P28482 1/20 0.32
CASP1 P29466 1/20 0.32
CASP7 P55210 1/20 0.32
DRD2 P14416 1/20 0.30
DRD3 P35462 1/20 0.30
NSD2 O96028 1/20 0.30
PABPC1 P11940 1/20 0.30
CSF1R P07333 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28499600 0.89 ALDH1A1 (0.39) KCNJ5KCNJ3LMNAALDH1A1HTR7
SCHEMBL427905 0.82 LMNA (0.45) LMNAALDH1A1KHKHTR7GAA
SCHEMBL28509585 0.78 ALDH1A1 (0.33) ALDH1A1GAAMEN1KMT2A
SCHEMBL28504600 0.77 LMNA (0.39) KCNJ5KCNJ3LMNAALDH1A1KHK
SCHEMBL28499619 0.77 DRD4 (0.40) KCNJ5KCNJ3LMNAALDH1A1KHK
SCHEMBL28502440 0.74 GAA (0.54) LMNAALDH1A1GAAMEN1KMT2A
SCHEMBL428655 0.74 ROCK1 (0.34) ALDH1A1MEN1KMT2AKDM4ETSHR
SCHEMBL24723411 0.73 LPL (0.33) ALDH1A1GAAMEN1KMT2AKDM4E
SCHEMBL586151 0.71 LPL (0.41) ALDH1A1GAAMEN1KMT2AKDM4E
SCHEMBL18621693 0.70 DRD2 (0.45) DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112243439-A Pyrrolo [2,3-B ] pyridines or pyrrolo [2,3-B ] pyrazines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-01-19 CN disclosed