SCHEMBL28501074

SCHEMBL28501074

C=C(C)c1cccc(C2=CCNCC2)n1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.42
HTR2C P28335 9/20 0.41
QDPR P09417 3/20 0.41
PIM1 P11309 1/20 0.40
PIM3 Q86V86 1/20 0.40
PIM2 Q9P1W9 1/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
HTR2A P28223 1/20 0.39
HTT P42858 1/20 0.39
RAD52 P43351 1/20 0.39
HTR6 P50406 1/20 0.39
CDK9 P50750 1/20 0.37
SCN9A Q15858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1942147 0.81 SIGMAR1 (0.47) SIGMAR1HTR2CQDPRPIM1PIM3
SCHEMBL7934174 0.80 SCN9A (0.40) SIGMAR1HTR2CQDPRPIM1PIM3
SCHEMBL171596 0.77 PIM1 (0.51) SIGMAR1HTR2CQDPRPIM1PIM3
SCHEMBL4294398 0.77 SCN9A (0.39) SIGMAR1HTR2CQDPRPIM1PIM3
SCHEMBL5341889 0.75 HTR2C (0.51) SIGMAR1HTR2CQDPRPIM1PIM3
SCHEMBL30454060 0.75 HTR2C (0.51) SIGMAR1HTR2CQDPRPIM1PIM3
SCHEMBL14761633 0.74 CDK9 (0.57) SIGMAR1HTR2CQDPRPIM1PIM3
SCHEMBL7940586 0.74 SIGMAR1 (0.49) SIGMAR1HTR2CQDPRPIM1PIM3
SCHEMBL3453255 0.74 HTR2C (0.51) SIGMAR1HTR2CQDPRPIM1PIM3
SCHEMBL13490658 0.74 SIGMAR1 (0.49) SIGMAR1HTR2CQDPRPIM1PIM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112119077-A Kinase inhibitors 曼彻斯特大学 2020-12-22 CN disclosed